SCHEMBL30132604

SCHEMBL30132604

COc1c(Oc2ccc(Cl)cc2)ccc2c1OCCC2N

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C19 P33261 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
SLC6A4 P31645 5/20 0.34
HTR2A P28223 4/20 0.34
KCNH2 Q12809 3/20 0.34
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
PTGDR2 Q9Y5Y4 7/20 0.33
SLC6A2 P23975 1/20 0.32
SLC6A3 Q01959 1/20 0.32
DPP4 P27487 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20554321 1.00 MAPT (0.35) MAPTKDM4EMEN1ALDH1A1CYP1A2
SCHEMBL30132559 0.85 MAPT (0.36) MAPTKDM4EMEN1ALDH1A1CYP1A2
SCHEMBL20554534 0.85 MAPT (0.36) MAPTKDM4EMEN1ALDH1A1CYP1A2
SCHEMBL20554267 0.85 HTR2A (0.33) HPGDKMT2ASLC6A4HTR2AHTR2C
SCHEMBL30132527 0.85 HTR2A (0.33) HPGDKMT2ASLC6A4HTR2AHTR2C
SCHEMBL20554109 0.85 L3MBTL1 (0.41) MAPTKDM4ESLC6A4HTR2AKCNH2
SCHEMBL30132635 0.82 MAPT (0.36) MAPTKDM4EMEN1ALDH1A1CYP1A2
SCHEMBL20554374 0.82 MAPT (0.36) MAPTKDM4EMEN1ALDH1A1CYP1A2
SCHEMBL20554813 0.78 ALOX5AP (0.39)
SCHEMBL20554695 0.76 PTGDR2 (0.35) PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110770211-B Alpha, beta unsaturated amide compound 协和麒麟株式会社 2023-09-19 CN disclosed
CN-108430972-B Alpha, beta-unsaturated amide compound 协和麒麟株式会社 2022-12-27 CN disclosed