SCHEMBL30132701

SCHEMBL30132701

NC1COc2cccc(Oc3ccc(C(F)(F)F)cc3)c2C1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.35
SCN9A Q15858 3/20 0.34
KCNH2 Q12809 2/20 0.34
SCN5A Q14524 2/20 0.34
L3MBTL1 Q9Y468 3/20 0.34
RAB9A P51151 1/20 0.34
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
DRD1 P21728 1/20 0.33
HTR1B P28222 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33
LTA4H P09960 1/20 0.33
MAPT P10636 2/20 0.32
LMNA P02545 1/20 0.32
ATM Q13315 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20554071 1.00 TRPV1 (0.35) TRPV1SCN9AKCNH2SCN5AL3MBTL1
SCHEMBL30132647 0.83 HTT (0.37) HTR1ADRD2DRD1HTR1BHTR2A
SCHEMBL20554767 0.83 HTT (0.37) HTR1ADRD2DRD1HTR1BHTR2A
SCHEMBL20554318 0.80 DRD2 (0.41) TRPV1SCN9AL3MBTL1RAB9ADRD2
SCHEMBL19054515 0.75 TEAD1 (0.50) SCN9AKCNH2SCN5AMTNR1A
SCHEMBL30132586 0.75 TEAD1 (0.50) SCN9AKCNH2SCN5AMTNR1A
SCHEMBL873501 0.74 DRD2 (0.54) HTR1ADRD2DRD1HTR1BHTR2A
SCHEMBL4839911 0.74 DRD2 (0.54) HTR1ADRD2DRD1HTR1BHTR2A
SCHEMBL873500 0.74 DRD2 (0.54) HTR1ADRD2DRD1HTR1BHTR2A
SCHEMBL19667511 0.68 KDM1A (0.44) L3MBTL1HTR1AHTR2CLTA4HMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110770211-B Alpha, beta unsaturated amide compound 协和麒麟株式会社 2023-09-19 CN disclosed
CN-108430972-B Alpha, beta-unsaturated amide compound 协和麒麟株式会社 2022-12-27 CN disclosed