SCHEMBL30135971

SCHEMBL30135971

CCCCOC(=O)N1CC2(CCC(NC(=O)c3ccc(Nc4ncc5c(n4)N(C4CCCC4)CC(F)(F)C(=O)N5C)c(OC)c3)CC2)C1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 18/20 0.72
BRD4 O60885 3/20 0.72
BRDT Q58F21 3/20 0.72
PLK3 Q9H4B4 4/20 0.57
PLK2 Q9NYY3 2/20 0.57
PRKD3 O94806 1/20 0.57
MAP4K4 O95819 1/20 0.57
PRKCG P05129 1/20 0.57
CLK2 P49760 1/20 0.57
RPS6KA3 P51812 1/20 0.57
NEK4 P51957 1/20 0.57
PTK2 Q05397 1/20 0.57
CAMK2G Q13555 1/20 0.57
CAMK2D Q13557 1/20 0.57
SRPK1 Q96SB4 1/20 0.57
PRKD2 Q9BZL6 1/20 0.57
CSNK1G1 Q9HCP0 1/20 0.57
CSNK1G3 Q9Y6M4 1/20 0.57
ALK Q9UM73 1/20 0.57
RAD52 P43351 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30135796 0.94 PLK1 (0.79) PLK1BRD4BRDTPLK3PLK2
SCHEMBL30135711 0.92 PLK1 (0.71) PLK1BRD4BRDTPLK3PLK2
SCHEMBL30135781 0.88 PLK1 (0.67) PLK1BRD4BRDTPLK3PLK2
SCHEMBL30136097 0.87 PLK1 (0.67) PLK1BRD4BRDTPLK3PLK2
SCHEMBL12330693 0.87 PLK1 (0.92) PLK1BRD4BRDTPLK3PLK2
SCHEMBL1559771 0.87 PLK1 (0.92) PLK1BRD4BRDTPLK3PLK2
SCHEMBL1559612 0.87 PLK1 (0.92) PLK1BRD4BRDTPLK3PLK2
SCHEMBL30135787 0.87 PLK1 (0.81) PLK1BRD4BRDTPLK3PLK2
SCHEMBL1675854 0.86 PLK1 (0.90) PLK1BRD4BRDTPLK3PLK2
SCHEMBL30135947 0.85 PLK1 (0.63) PLK1BRD4BRDTPLK3PLK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4384520-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND Uppthera, Inc. (KR) 2024-06-19 EP disclosed
WO-2023017446-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND UPPTHERA, INC. (KR) 2023-02-16 WO disclosed
WO-2023017442-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND UPPTHERA, INC. (KR) 2023-02-16 WO disclosed