SCHEMBL30139729

SCHEMBL30139729

Nc1ncc2c(N)nn(-c3ccc(N4CCNCC4)nc3)c2n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.45
GPR119 Q8TDV5 1/20 0.38
HRH4 Q9H3N8 2/20 0.38
CHRNB2 P17787 2/20 0.37
CHRNA4 P43681 2/20 0.37
ATR Q13535 1/20 0.37
OPRM1 P35372 1/20 0.36
OPRL1 P41146 1/20 0.36
AXL P30530 3/20 0.36
MERTK Q12866 3/20 0.36
PLD1 Q13393 1/20 0.36
TYRO3 Q06418 1/20 0.36
ITGA2B P08514 1/20 0.36
AURKA O14965 2/20 0.36
RET P07949 2/20 0.36
KIT P10721 2/20 0.36
SRC P12931 2/20 0.36
KDR P35968 2/20 0.36
FLT3 P36888 2/20 0.36
MET P08581 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL30139731 0.90 CHRNB2 (0.42) HRH3HRH4CHRNB2CHRNA4
SCHEMBL30139795 0.86 HRH3 (0.47) HRH3HRH4ATRPTPN11
SCHEMBL30139759 0.72 TLR9 (0.38) HRH3AXLMERTKTYRO3AURKA
SCHEMBL23711942 0.71 PARP1 (0.42)
SCHEMBL30139810 0.71 KHK (0.46) ATRTBK1
SCHEMBL30139792 0.71 PARP1 (0.42)
SCHEMBL4753475 0.71 EGFR (0.49) SRC
SCHEMBL31347924 0.68 PLD1 (0.53) HRH3GPR119HRH4CHRNB2CHRNA4
SCHEMBL529383 0.68 PLD1 (0.53) HRH3GPR119HRH4CHRNB2CHRNA4
Hydrochloric Acid SCHEMBL25317270 0.67 CHRNB2 (0.60) GPR119HRH4CHRNB2CHRNA4PLD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022270994-A1 NOVEL BIFUNCTIONAL HETEROCYCLIC COMPOUND HAVING BTK DEGRADATION FUNCTION VIA UBIQUITIN PROTEASOME PATHWAY, AND USE THEREOF 한국화학연구원 2022-12-29 WO disclosed