SCHEMBL30140677

SCHEMBL30140677

Cc1nc(N2CC3CC3C2)ncc1CN=[N+]=[N-]

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 6/20 0.36
RBP4 P02753 2/20 0.35
DYRK1A Q13627 1/20 0.33
HCRTR1 O43613 4/20 0.32
HCRTR2 O43614 4/20 0.32
CHRM4 P08173 1/20 0.31
PDE5A O76074 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21747035 1.00 KLKB1 (0.36) KLKB1RBP4DYRK1AHCRTR1HCRTR2
SCHEMBL21747131 0.84 KLKB1 (0.36) KLKB1
SCHEMBL30140673 0.84 KLKB1 (0.36) KLKB1
SCHEMBL23469510 0.78 KLKB1 (0.41) KLKB1RBP4DYRK1AHCRTR1HCRTR2
SCHEMBL20541008 0.78 NR1H2 (0.45) KLKB1RBP4DYRK1AHCRTR1HCRTR2
SCHEMBL18794997 0.78 HDAC3 (0.33) RBP4
SCHEMBL21746998 0.78 KLKB1 (0.39) KLKB1
SCHEMBL21736743 0.69 KLKB1 (0.49) KLKB1RBP4HCRTR1HCRTR2
SCHEMBL21736872 0.66 KLKB1 (0.47) KLKB1RBP4HCRTR1HCRTR2
SCHEMBL22166243 0.66 KLKB1 (0.59) KLKB1RBP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113039181-B Heteroaromatic carboxamide derivatives as inhibitors of plasma kallikrein 勃林格殷格翰国际有限公司 2024-08-13 CN disclosed
CN-110546146-B Heteroaryl carboxamide derivatives as plasma kallikrein inhibitors 勃林格殷格翰国际有限公司 2023-02-21 CN disclosed