SCHEMBL30140692

SCHEMBL30140692

O=C1c2ccccc2C(=O)N1c1cccnc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 1.00
GAA P10253 2/20 0.73
MAPT P10636 2/20 0.73
HSD17B10 Q99714 2/20 0.73
MAPK1 P28482 1/20 0.73
KDM4E B2RXH2 3/20 0.60
CYP11B2 P19099 1/20 0.57
FFAR4 Q5NUL3 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.54
ALDH1A1 P00352 3/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
ELANE P08246 1/20 0.51
AR P10275 1/20 0.50
IDO1 P14902 1/20 0.49
TDO2 P48775 1/20 0.49
RECQL P46063 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
RAB9A P51151 1/20 0.47
CCR9 P51686 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22668259 0.87 HTT (0.77) HTTGAAMAPTHSD17B10MAPK1
SCHEMBL18589024 0.84 HTT (0.73) HTTGAAMAPTHSD17B10MAPK1
SCHEMBL4122353 0.82 HTT (0.70) HTTGAAMAPTHSD17B10MAPK1
SCHEMBL441164 0.82 HTT (0.70) HTTGAAMAPTHSD17B10MAPK1
SCHEMBL16862943 0.82 HTT (0.69) HTTGAAMAPTHSD17B10MAPK1
SCHEMBL16862998 0.81 HTT (0.67) HTTGAAMAPTHSD17B10MAPK1
SCHEMBL29644725 0.80 HTT (0.67) HTTGAAMAPTHSD17B10MAPK1
SCHEMBL28603975 0.80 HTT (0.67) HTTGAAMAPTHSD17B10MAPK1
SCHEMBL11619942 0.78 KDM4E (0.70) HTTGAAKDM4EALDH1A1SMN1; SMN2
N-Phenyl-Phthalimide SCHEMBL29819622 0.77 KMT2A (0.68) HTTGAAMAPTHSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110546146-B Heteroaryl carboxamide derivatives as plasma kallikrein inhibitors 勃林格殷格翰国际有限公司 2023-02-21 CN disclosed