SCHEMBL30142489

SCHEMBL30142489

COc1ccc2c(c1)CN(C(N)=O)C2

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RYR2 Q92736 7/20 0.62
ESR1 P03372 1/20 0.56
ESR2 Q92731 1/20 0.56
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA7 P43166 1/20 0.52
CA9 Q16790 1/20 0.52
CA14 Q9ULX7 1/20 0.52
HSD17B10 Q99714 1/20 0.51
ABHD6 Q9BV23 1/20 0.50
HSP90AA1 P07900 1/20 0.50
NAMPT P43490 3/20 0.48
TAS1R3 Q7RTX0 1/20 0.47
TAS1R1 Q7RTX1 1/20 0.47
TAS1R2 Q8TE23 1/20 0.47
ROCK1 Q13464 2/20 0.46
TMPRSS2 O15393 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15880544 0.85 ESR1 (0.57) RYR2ESR1ESR2CA1CA2
SCHEMBL30677763 0.85 ESR1 (0.57) RYR2ESR1ESR2CA1CA2
SCHEMBL14590586 0.85 ESR1 (0.57) RYR2ESR1ESR2CA1CA2
SCHEMBL16282723 0.81 ESR1 (0.60) RYR2ESR1ESR2CA1CA2
SCHEMBL15989340 0.81 ESR1 (0.53) RYR2ESR1ESR2CA1CA2
SCHEMBL17341937 0.81 NAMPT (0.53) RYR2ESR1ESR2CA1CA2
SCHEMBL25825941 0.80 ESR1 (0.80) RYR2ESR1ESR2CA1CA2
SCHEMBL30685013 0.80 ESR1 (0.52) RYR2ESR1ESR2CA1CA2
SCHEMBL24761144 0.78 ESR2 (0.56) ESR1ESR2CA1CA2CA7
SCHEMBL6234508 0.78 ESR1 (0.51) RYR2ESR1ESR2CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109843379-B Substituted ureas and methods of making and using the same 梅比斯发现公司 2022-12-30 CN disclosed