SCHEMBL30142914

SCHEMBL30142914

CON(C)C(=O)C[C@@H](C)c1c(I)ncnc1N1CCNCC1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 4/20 0.36
USP2 O75604 3/20 0.36
TSHR P16473 2/20 0.36
HSD17B10 Q99714 2/20 0.36
CYP2D6 P10635 2/20 0.36
ENPP1 P22413 1/20 0.36
HTR2C P28335 5/20 0.33
CYP1A2 P05177 3/20 0.33
CYP3A4 P08684 3/20 0.33
CYP2C19 P33261 3/20 0.33
MAPT P10636 2/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
ALDH1A1 P00352 1/20 0.31
DRD2 P14416 1/20 0.31
CSNK1A1 P48729 2/20 0.31
TLR7 Q9NYK1 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28337228 0.88 MAPT (0.33) TSHRENPP1HTR2CMAPT
SCHEMBL28339340 0.87 AURKA (0.35) TSHRENPP1MAPTKDM4EHPGD
SCHEMBL28339341 0.87 AURKA (0.35) TSHRENPP1MAPTKDM4EHPGD
SCHEMBL16773148 0.85 AURKA (0.30)
SCHEMBL15389848 0.85 ENPP1 (0.38) CLK4USP2TSHRHSD17B10CYP2D6
SCHEMBL15390257 0.83 AURKA (0.41) CLK4USP2TSHRHSD17B10CYP2D6
SCHEMBL21485106 0.78 LIMK2 (0.35)
SCHEMBL21485105 0.78 LIMK2 (0.35)
SCHEMBL16755390 0.69 KIT (0.47) KDM4ETLR7
SCHEMBL16773364 0.69 AURKA (0.41) USP2TSHRHSD17B10CYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110590606-B Process for preparing pyrimidylcyclopentane compounds 豪夫迈·罗氏有限公司 2023-02-17 CN disclosed