SCHEMBL30145264

SCHEMBL30145264

Cc1c(Br)cccc1-c1nc2c(o1)CN(C(=O)OCc1ccccc1)C2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.40
PARP2 Q9UGN5 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
PDCD1 Q15116 6/20 0.39
CD274 Q9NZQ7 6/20 0.39
PTGDR2 Q9Y5Y4 3/20 0.38
TMEM97 Q5BJF2 2/20 0.38
SIGMAR1 Q99720 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
GRM5 P41594 1/20 0.38
HTR1A P08908 1/20 0.38
ADRA2A P08913 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38
DRD1 P21728 1/20 0.38
HRH2 P25021 1/20 0.38
HTR1B P28222 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20293305 1.00 PARP1 (0.40) PARP1PARP2MEN1KMT2ANPSR1
SCHEMBL20296159 0.92 PTGDR2 (0.45) MEN1KMT2ANPSR1PTGDR2TMEM97
SCHEMBL30740274 0.92 PTGDR2 (0.45) MEN1KMT2ANPSR1PTGDR2TMEM97
SCHEMBL14991147 0.80 MEN1 (0.49) PARP1PARP2MEN1KMT2ANPSR1
SCHEMBL20293210 0.80 PDCD1 (0.42) PDCD1CD274
SCHEMBL20293007 0.78 PDCD1 (0.53) PDCD1CD274
SCHEMBL17982156 0.77 S1PR5 (0.46) MEN1KMT2ANPSR1PTGDR2GRM5
SCHEMBL505281 0.77 GRM5 (0.48) MEN1KMT2ANPSR1CYP3A4GRM5
SCHEMBL30740215 0.77 PDCD1 (0.52) PDCD1CD274
SCHEMBL20296086 0.77 PDCD1 (0.51) PDCD1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110267953-B Tetrahydroimidazo [4,5-C ] pyridine derivatives as inducers of PD-L1 internalization 因赛特公司 2022-12-20 CN disclosed