SCHEMBL30740274

SCHEMBL30740274

Cc1c(Br)cccc1-c1nc2c(o1)CCN(C(=O)OCc1ccccc1)C2

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 7/20 0.45
TMEM97 Q5BJF2 4/20 0.44
SIGMAR1 Q99720 4/20 0.44
GRM5 P41594 3/20 0.43
S1PR5 Q9H228 2/20 0.43
KDR P35968 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
DHFR P00374 1/20 0.42
PPARA Q07869 1/20 0.42
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20296159 1.00 PTGDR2 (0.45) PTGDR2TMEM97SIGMAR1GRM5S1PR5
SCHEMBL20293305 0.92 PARP1 (0.40) PTGDR2TMEM97SIGMAR1GRM5S1PR5
SCHEMBL30145264 0.92 PARP1 (0.40) PTGDR2TMEM97SIGMAR1GRM5S1PR5
SCHEMBL505382 0.81 PPARA (0.50) PTGDR2TMEM97SIGMAR1GRM5S1PR5
SCHEMBL17377166 0.81 DHFR (0.49) PTGDR2TMEM97SIGMAR1GRM5KDR
SCHEMBL504679 0.79 S1PR5 (0.52) TMEM97SIGMAR1GRM5S1PR5KDR
SCHEMBL504584 0.79 DHFR (0.44) PTGDR2TMEM97SIGMAR1GRM5S1PR5
SCHEMBL505215 0.78 GRM5 (0.56) GRM5S1PR5DHFR
SCHEMBL504656 0.78 DHFR (0.46) PTGDR2TMEM97SIGMAR1GRM5KDR
SCHEMBL10250503 0.78 DHFR (0.48) PTGDR2TMEM97SIGMAR1GRM5S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110582493-B Benzoxazole derivatives as immunomodulators 因赛特公司 2024-03-08 CN disclosed