SCHEMBL301454

SCHEMBL301454

CCC(O)OC(=O)/C=C/C(=O)OC(O)CC

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.43
HCAR2 Q8TDS4 9/20 0.43
ATM Q13315 1/20 0.38
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
GAPDH P04406 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL950768 1.00 TSHR (0.43) TSHRHCAR2ATMKEAP1NFE2L2
SCHEMBL301455 1.00 TSHR (0.43) TSHRHCAR2ATMKEAP1NFE2L2
SCHEMBL950770 0.91 HCAR2 (0.57) TSHRHCAR2ATMKEAP1NFE2L2
SCHEMBL769452 0.91 HCAR2 (0.57) TSHRHCAR2ATMKEAP1NFE2L2
SCHEMBL28178149 0.91 HCAR2 (0.54) TSHRHCAR2ATMKEAP1NFE2L2
SCHEMBL8417690 0.91 HCAR2 (0.54) TSHRHCAR2ATMKEAP1NFE2L2
SCHEMBL8641563 0.91 HCAR2 (0.57) TSHRHCAR2ATMKEAP1NFE2L2
SCHEMBL8641572 0.91 HCAR2 (0.57) TSHRHCAR2ATMKEAP1NFE2L2
SCHEMBL27660385 0.91 HCAR2 (0.57) TSHRHCAR2ATMKEAP1NFE2L2
SCHEMBL8417684 0.91 HCAR2 (0.54) TSHRHCAR2ATMKEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5733951-A ESTER INTERCHANGE OF BIS/HYDROXYPROPYL/ FUMARATE WM. MARSH RICE UNIVERSITY 1998-03-31 US claimed
WO-1995029710-A1 POLY(PROPYLENE FUMARATE) RICE UNIVERSITY (US) 1995-11-09 WO claimed
EP-3576802-B1 A THERMORESPONSIVE HYDROGEL UNIV JOHANNESBURG WITWATERSRAND (ZA) 2022-06-29 EP disclosed
US-11197948-B2 Thermoresponsive hydrogel UNIVERSITY OF THE WITWATERSRAND, JOHANNESBURG (ZA) 2021-12-14 US disclosed
US-20200054791-A1 A Thermoresponsive Hydrogel UNIVERSITY OF THE WITWATERSRAND, JOHANNESBURG (ZA) 2020-02-20 US disclosed
WO-2018142299-A1 A THERMORESPONSIVE HYDROGEL UNIVERSITY OF THE WITWATERSRAND, JOHANNESBURG (ZA) 2018-08-09 WO disclosed
US-9795471-B2 Polymer-tissue hybrid biomaterials and methods of making and using same UNIVERSITY OF MARYLAND, COLLEGE PARK (US) 2017-10-24 US disclosed
US-20160089476-A1 POLYMER-TISSUE HYBRID BIOMATERIALS AND METHODS OF MAKING AND USING SAME NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2016-03-31 US disclosed
EP-1812481-B1 BLOCK COPOLYMERS OF POLYCAPROLACTONE AND POLY (PROPYLENE FUMARATE) MAYO FOUNDATION (US) 2012-01-11 EP disclosed
EP-1409566-B1 PHOTOCROSSLINKING OF DIETHYL FUMARATE/POLY(PROPYLENE FUMARATE) BIOMATERIALS UNIV WM MARSH RICE (US) 2008-04-23 EP disclosed
EP-1812481-A2 BLOCK COPOLYMERS OF POLYCAPROLACTONE AND POLY (PROPYLENE FUMARATE) Mayo Foundation for Medical Education and Research (US) 2007-08-01 EP disclosed
US-6753358-B2 POLYMER NETWORK COMPRISING POLY(PROPYLENE FUMARATE) CROSSLINKED WITH A FUMARATE DERIVATIVE SUCH AS DIETHYL FUMARATE; BIODEGRADABLE; USEFUL FOR IN VIVO APPLICATIONS; INJECTABLE; FOR RECONSTRUCTING BONE WILLIAM MARSH RICE UNIVERSITY 2004-06-22 US disclosed
EP-1409566-A2 PHOTOCROSSLINKING OF DIETHYL FUMARATE/POLY(PROPYLENE FUMARATE) BIOMATERIALS Wm. MARSH RICE UNIVERSITY (US) 2004-04-21 EP disclosed
US-20030032733-A1 Photocrosslinking of diethyl fumarate/poly (propylene fumarate) biomaterials WM. MARSH RICE UNIVERSITY (US) 2003-02-13 US disclosed
WO-2003002490-A2 PHOTOCROSSLINKING OF DIETHYL FUMARATE/POLY(PROPYLENE FUMARATE) BIOMATERIALS WM. MARSH RICE UNIVERSITY (US) 2003-01-09 WO disclosed
US-5733951-A ESTER INTERCHANGE OF BIS/HYDROXYPROPYL/ FUMARATE WM. MARSH RICE UNIVERSITY 1998-03-31 US disclosed
WO-1995029710-A1 POLY(PROPYLENE FUMARATE) RICE UNIVERSITY (US) 1995-11-09 WO disclosed
US-4151149-A OXYGEN BARRIER MEMBRANES, SULFATED MONOMERS UNION OIL COMPANY OF CALIFORNIA (US) 1979-04-24 US disclosed
US-4079025-A ADDITION POLYMER A. E. STALEY MANUFACTURING COMPANY (US) 1978-03-14 US disclosed
US-4007141-A Opaque, non-pigmented microporous film and process and composition for preparing same PPG INDUSTRIES, INC. (US) 1977-02-08 US disclosed