SCHEMBL30147733

SCHEMBL30147733

CCOC(=O)c1cnn(-c2cncc(C#N)c2)c1C(F)(F)F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPC1 P48995 2/20 0.52
TRPC3 Q13507 2/20 0.52
STIM1 Q13586 2/20 0.52
ORAI1 Q96D31 2/20 0.52
STIM2 Q9P246 2/20 0.52
HPGD P15428 7/20 0.49
ALDH1A1 P00352 7/20 0.49
KDM4E B2RXH2 6/20 0.49
MAPT P10636 5/20 0.49
L3MBTL1 Q9Y468 4/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
GAA P10253 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
CYP1A2 P05177 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
POLB P06746 1/20 0.45
MALT1 Q9UDY8 2/20 0.44
GUCY1A1 Q02108 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21604844 1.00 TRPC1 (0.52) TRPC1TRPC3STIM1ORAI1STIM2
SCHEMBL31252546 0.86 KDM4E (0.56) TRPC1TRPC3STIM1ORAI1STIM2
SCHEMBL6180211 0.86 KDM4E (0.56) TRPC1TRPC3STIM1ORAI1STIM2
SCHEMBL1402810 0.86 TRPC1 (0.62) TRPC1TRPC3STIM1ORAI1STIM2
SCHEMBL30147621 0.85 TRPC1 (0.56) TRPC1TRPC3STIM1ORAI1STIM2
SCHEMBL21604958 0.85 TRPC1 (0.56) TRPC1TRPC3STIM1ORAI1STIM2
SCHEMBL30147292 0.82 MALT1 (0.48) ALDH1A1KDM4EMAPTTDP1POLB
SCHEMBL21604960 0.82 TRPC1 (0.59) TRPC1TRPC3STIM1ORAI1STIM2
SCHEMBL21604941 0.80 KDM4E (0.51) TRPC1TRPC3STIM1ORAI1STIM2
SCHEMBL30147895 0.80 KDM4E (0.51) TRPC1TRPC3STIM1ORAI1STIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112585128-B Pyrazole derivatives as MALT1 inhibitors 詹森药业有限公司 2023-02-21 CN disclosed