SCHEMBL6180211

SCHEMBL6180211

CCOC(=O)c1cnn(-c2cccc(C#N)c2)c1C(F)(F)F

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.56
ALDH1A1 P00352 8/20 0.56
HPGD P15428 7/20 0.56
MAPT P10636 6/20 0.56
TRPC1 P48995 2/20 0.53
TRPC3 Q13507 2/20 0.53
STIM1 Q13586 2/20 0.53
ORAI1 Q96D31 2/20 0.53
STIM2 Q9P246 2/20 0.53
L3MBTL1 Q9Y468 4/20 0.52
MEN1 O00255 2/20 0.52
GAA P10253 2/20 0.52
KMT2A Q03164 2/20 0.52
CYP1A2 P05177 2/20 0.52
CYP2C9 P11712 2/20 0.52
CYP2C19 P33261 2/20 0.52
HTT P42858 2/20 0.51
TDP1 Q9NUW8 1/20 0.51
POLB P06746 2/20 0.48
GUCY1A1 Q02108 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31252546 1.00 KDM4E (0.56) KDM4EALDH1A1HPGDMAPTTRPC1
SCHEMBL1402810 0.87 TRPC1 (0.62) KDM4EALDH1A1HPGDMAPTTRPC1
SCHEMBL30147733 0.86 TRPC1 (0.52) KDM4EALDH1A1HPGDMAPTTRPC1
SCHEMBL21604844 0.86 TRPC1 (0.52) KDM4EALDH1A1HPGDMAPTTRPC1
SCHEMBL18706884 0.84 KDM4E (0.56) KDM4EALDH1A1HPGDMAPTTRPC1
SCHEMBL31117196 0.84 HTT (0.72) KDM4EALDH1A1HPGDMAPTMEN1
SCHEMBL4161763 0.84 HTT (0.72) KDM4EALDH1A1HPGDMAPTMEN1
SCHEMBL26125572 0.83 MAPT (0.67) KDM4EALDH1A1MAPTKMT2ATDP1
SCHEMBL31252567 0.83 MAPT (0.67) KDM4EALDH1A1MAPTKMT2ATDP1
SCHEMBL21604941 0.83 KDM4E (0.51) KDM4EALDH1A1HPGDMAPTTRPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4707276-A2 MALT1 MODULATORS AND USES THEREOF Rarefied Biosciences, Inc. (US) 2026-03-11 EP disclosed
EP-4499611-B1 MALT1 MODULATORS AND USES THEREOF RAREFIED BIOSCIENCES INC (US) 2026-02-18 EP disclosed
US-20250326738-A1 MALT1 Modulators and Uses Thereof RAREFIED BIOSCIENCES, INC. (US) 2025-10-23 US disclosed
EP-4499611-A1 MALT1 MODULATORS AND USES THEREOF Rarefied Biosciences, Inc. (US) 2025-02-05 EP disclosed
CN-119032083-A MALT1 modulators and uses thereof 稀有生物科学股份有限公司 2024-11-26 CN disclosed
WO-2023192506-A1 MALT1 MODULATORS AND USES THEREOF RARIFIED BIOSCIENCES, INC. (US) 2023-10-05 WO disclosed
US-20050239797-A1 Isoquinoline and quinazoline derivatives having a combined 5HT1A, 5HT1B, and 5HT1D receptor activity SMITHKLINE BEECHAM, PLC 2005-10-27 US disclosed
EP-1228043-B1 ISOQUINOLINE AND QUINAZOLINE DEIVATIVES HAVING A COMBINED 5HT1A, 5HT1B AND 5HT1D RECEPTOR ACTIVITY SMITHKLINE BEECHAM PLC (GB) 2005-01-12 EP disclosed
EP-1228043-A1 ISOQUINOLINE AND QUINAZOLINE DEIVATIVES HAVING A COMBINED 5HT1A, 5HT1B AND 5HT1D RECEPTOR ACTIVITY SMITHKLINE BEECHAM PLC (GB) 2002-08-07 EP disclosed
WO-2001032626-A1 ISOQUINOLINE AND QUINAZOLINE DERIVATIVES HAVING A COMBINED 5HT1A, 5HT1B AND 5HT1D RECEPTOR ACTIVITY SMITHKLINE BEECHAM P.L.C. (GB) 2001-05-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250326738-A1 MALT1 Modulators and Uses Thereof MALT1, SQSTM1, PPP1R10 KDM4E 2044/4885ALDH1A1 3447/4885HPGD 3460/4885
US-20050239797-A1 Isoquinoline and quinazoline derivatives having a combined 5HT1A, 5HT1B, and 5HT1D receptor activity HTR1B, HTR1A, HTR1D KDM4E 3839/4885ALDH1A1 489/4885HPGD 1763/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.