SCHEMBL30152003

SCHEMBL30152003

O=C(Nc1ccc2c(cnn2Cc2ccccc2)c1)c1cnc(Nc2cccc(NCCCn3ccnc3)n2)s1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 6/20 0.51
EGFR P00533 5/20 0.51
LCK P06239 2/20 0.44
KIT P10721 1/20 0.40
BRAF P15056 1/20 0.40
NAMPT P43490 1/20 0.39
FGFR1 P11362 1/20 0.39
SRC P12931 1/20 0.39
ITGB3 P05106 5/20 0.39
ITGAV P06756 5/20 0.39
ITGA2B P08514 4/20 0.39
ALDH1A1 P00352 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.37
HTT P42858 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL774573 1.00 ERBB2 (0.51) ERBB2EGFRLCKKITBRAF
SCHEMBL773111 0.88 EGFR (0.50) ERBB2EGFRKITBRAFFGFR1
SCHEMBL30151993 0.88 EGFR (0.50) ERBB2EGFRKITBRAFFGFR1
SCHEMBL774604 0.86 LCK (0.50) EGFRLCKKITBRAFNAMPT
SCHEMBL773549 0.83 LCK (0.52) LCKNAMPTALDH1A1L3MBTL1
SCHEMBL774920 0.82 LCK (0.47) LCKNAMPTALDH1A1KDM4ELMNA
SCHEMBL774149 0.80 LCK (0.55) LCKNAMPTFGFR1SRCALDH1A1
SCHEMBL774538 0.80 ALDH1A1 (0.51) LCKNAMPTALDH1A1KDM4ELMNA
SCHEMBL774389 0.79 LCK (0.55) EGFRLCKNAMPTALDH1A1L3MBTL1
SCHEMBL773381 0.78 LCK (0.49) LCKKITBRAFNAMPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4139305-A1 HALOGENATED-HETEROARYL AND OTHER HETEROCYCLIC KINASE INHIBITORS, AND USES THEREOF iOmx Therapeutics AG (DE) 2023-03-01 EP disclosed