SCHEMBL30159633

SCHEMBL30159633

COC(=O)c1ccc2[nH]nc(C)c2c1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
CASP3 P42574 1/20 0.43
SENP8 Q96LD8 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
SENP6 Q9GZR1 1/20 0.43
MAPT P10636 2/20 0.41
KDM4E B2RXH2 3/20 0.40
STAT3 P40763 1/20 0.40
HIF1A Q16665 1/20 0.40
MAP2K4 P45985 1/20 0.39
NR4A2 P43354 5/20 0.38
AR P10275 1/20 0.38
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23535659 1.00 NPC1 (0.43) NPC1RAB9ASMN1; SMN2CASP3SENP8
SCHEMBL2864348 0.84 NR4A2 (0.40) NPC1RAB9ASMN1; SMN2CASP3SENP8
SCHEMBL23535768 0.83 TTR (0.43) SMN1; SMN2KDM4EMAP2K4TTR
SCHEMBL1394029 0.79 MAPT (0.49) MAPTKDM4ESTAT3HIF1ANR4A2
SCHEMBL27536113 0.76 MAP2K4 (0.47) MAP2K4LRRK2KDR
SCHEMBL4150250 0.75 CHEK1 (0.43) NPC1RAB9ASMN1; SMN2MAPTMAP2K4
SCHEMBL4150252 0.75 CHEK1 (0.43) NPC1RAB9ASMN1; SMN2MAPTMAP2K4
SCHEMBL16759813 0.75 KDM4E (0.41) NPC1RAB9ASMN1; SMN2CASP3SENP8
SCHEMBL2867525 0.74 ALPL (0.50) SMN1; SMN2MAP2K4NR4A2CA12KDR
SCHEMBL522062 0.73 CA12 (0.52) NPC1RAB9ASMN1; SMN2CASP3SENP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4076440-A1 INHIBITORS OF ENL/AF9 YEATS The Rockefeller University (US) 2022-10-26 EP disclosed