SCHEMBL30161698

SCHEMBL30161698

CC(C)(C)OC(=O)N1CC(C(C)(C)Oc2cc(Br)cc3c2cnn3C2CCCCO2)C1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.37
TDO2 P48775 1/20 0.37
USP30 Q70CQ3 3/20 0.36
KRAS P01116 1/20 0.36
PDE4B Q07343 8/20 0.35
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
RXRG P48443 1/20 0.35
EHMT2 Q96KQ7 1/20 0.34
CCNK O75909 1/20 0.34
CDK12 Q9NYV4 1/20 0.34
EPHA2 P29317 1/20 0.33
ATR Q13535 3/20 0.33
PIK3CA P42336 1/20 0.33
MTOR P42345 1/20 0.33
PIK3CG P48736 1/20 0.33
AURKB Q96GD4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20699329 1.00 IDO1 (0.37) IDO1TDO2USP30KRASPDE4B
SCHEMBL30161639 0.90 SCN9A (0.36) USP30KRASPDE4BRXRARXRB
SCHEMBL20699301 0.90 SCN9A (0.36) USP30KRASPDE4BRXRARXRB
SCHEMBL20699309 0.86 SCN9A (0.41) IDO1TDO2USP30KRASPDE4B
SCHEMBL30161443 0.86 SCN9A (0.41) IDO1TDO2USP30KRASPDE4B
SCHEMBL20711762 0.84 PDE4B (0.43) IDO1TDO2USP30PDE4BCCNK
SCHEMBL29607485 0.84 PDE4B (0.43) IDO1TDO2USP30PDE4BCCNK
SCHEMBL28385243 0.84 PDE4B (0.43) IDO1TDO2USP30PDE4BCCNK
SCHEMBL20711872 0.83 RXRA (0.34) IDO1TDO2RXRARXRBRXRG
SCHEMBL20711770 0.82 KRAS (0.39) KRASPDE4BRXRARXRBRXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111032646-B Pyrazolo and triazolo bicyclic compounds as JAK kinase inhibitors 施万生物制药研发IP有限责任公司 2023-01-03 CN disclosed