SCHEMBL30161875

SCHEMBL30161875

CC(C)(Oc1cc(-c2ccc(O)cc2)nc2[nH]ncc12)C1CNC1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
FGFR1 P11362 1/20 0.34
FGFR2 P21802 1/20 0.34
FGFR3 P22607 1/20 0.34
GSK3B P49841 3/20 0.33
GSK3A P49840 2/20 0.33
CDK2 P24941 1/20 0.33
ALK Q9UM73 3/20 0.33
PIK3CA P42336 2/20 0.33
PIK3CD O00329 1/20 0.33
PIM1 P11309 1/20 0.33
PIK3CB P42338 1/20 0.33
SGK1 O00141 9/20 0.33
JAK2 O60674 2/20 0.32
JAK1 P23458 2/20 0.32
TYK2 P29597 2/20 0.32
JAK3 P52333 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20699358 1.00 ESR1 (0.36) ESR1ESR2FGFR1FGFR2FGFR3
Trifluoroacetic Acid SCHEMBL29607409 0.92 ESR1 (0.34) ESR1ESR2GSK3BGSK3ACDK2
SCHEMBL30161563 0.83 IDO1 (0.38) GSK3BGSK3ACDK2PIK3CAPIK3CD
SCHEMBL20699371 0.83 IDO1 (0.38) GSK3BGSK3ACDK2PIK3CAPIK3CD
SCHEMBL20715202 0.82 ESR1 (0.34) ESR1ESR2GSK3BGSK3AALK
SCHEMBL20699365 0.82 JAK3 (0.39) JAK3
SCHEMBL20711756 0.80 SGK1 (0.33) ESR1ESR2GSK3BGSK3ACDK2
SCHEMBL20699342 0.78 SGK1 (0.41) ESR1ESR2FGFR1FGFR2FGFR3
SCHEMBL30161715 0.78 SGK1 (0.41) ESR1ESR2FGFR1FGFR2FGFR3
SCHEMBL17667703 0.76 GSK3B (0.37) ESR1ESR2FGFR1FGFR2FGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111032646-B Pyrazolo and triazolo bicyclic compounds as JAK kinase inhibitors 施万生物制药研发IP有限责任公司 2023-01-03 CN disclosed