SCHEMBL30165253

SCHEMBL30165253

CS(=O)(=O)c1nc(Oc2ccc(F)cc2)cc(OC(C(N)=O)C23CC4CC(CC(C4)C2)C3)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 14/20 0.38
FPR2 P25090 8/20 0.38
EPHX2 P34913 1/20 0.36
ENPP3 O14638 1/20 0.33
CA12 O43570 1/20 0.33
ENPP1 P22413 1/20 0.33
ENPP2 Q13822 1/20 0.33
CA9 Q16790 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
BCL2 P10415 1/20 0.33
BCL2L1 Q07817 1/20 0.33
MCL1 Q07820 1/20 0.33
ABL1 P00519 1/20 0.32
F2 P00734 1/20 0.32
F10 P00742 1/20 0.32
PRSS1 P07477 1/20 0.32
PRSS2 P07478 1/20 0.32
PRSS3 P35030 1/20 0.32
ST14 Q9Y5Y6 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23884144 1.00 SCN9A (0.38) SCN9AFPR2EPHX2ENPP3CA12
SCHEMBL23884195 0.86 MAPT (0.39) SCN9AFPR2EPHX2CYP1A2CYP2C19
SCHEMBL30165318 0.86 MAPT (0.39) SCN9AFPR2EPHX2CYP1A2CYP2C19
SCHEMBL23907992 0.75 EPHX2 (0.46) EPHX2
SCHEMBL23884164 0.74 SCN9A (0.32) SCN9A
SCHEMBL30165244 0.74 SCN9A (0.32) SCN9A
SCHEMBL30165200 0.73 CYP3A4 (0.33)
SCHEMBL30361601 0.72 SCN9A (0.41) SCN9AFPR2CYP1A2CYP2C19F2
SCHEMBL30165226 0.68 ALDH1A1 (0.35) EPHX2
SCHEMBL30165307 0.67 MAPT (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4125845-A1 NOVEL 2-PYRIMIDONE ANALOGS AS POTENT ANTIVIRAL AGENTS AGAINST ALPHAVIRUSES Southern Research Institute (US) 2023-02-08 EP disclosed