SCHEMBL30172153

SCHEMBL30172153

NC(=O)Cc1ccc(Cl)cc1OC[C@@H](O)CNC1CCN(Cc2ccc(Cl)cc2)CC1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.62
HRH1 P35367 4/20 0.50
CCR3 P51677 4/20 0.50
LMNA P02545 1/20 0.50
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
KDM4E B2RXH2 1/20 0.47
MITF O75030 1/20 0.47
ALDH1A1 P00352 1/20 0.47
MAPT P10636 1/20 0.47
MAPK1 P28482 1/20 0.47
HTT P42858 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
BCHE P06276 2/20 0.45
ACHE P22303 2/20 0.45
BACE1 P56817 2/20 0.45
SIGMAR1 Q99720 2/20 0.44
ATF4 P18848 2/20 0.43
CCR5 P51681 3/20 0.43
ADRB2 P07550 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5141124 0.88 ABCB11 (0.55) ABCB11HRH1CCR3LMNAMEN1
SCHEMBL3149898 0.86 ABCB11 (0.63) ABCB11HRH1CCR3LMNAMEN1
SCHEMBL3149904 0.86 ABCB11 (0.63) ABCB11HRH1CCR3LMNAMEN1
SCHEMBL3145540 0.85 ABCB11 (0.61) ABCB11HRH1CCR3LMNAMEN1
SCHEMBL3145527 0.85 ABCB11 (0.61) ABCB11HRH1CCR3LMNAMEN1
SCHEMBL1683017 0.82 ABCB11 (0.83) ABCB11HRH1CCR3LMNAMEN1
Trifluoroacetic Acid SCHEMBL3145177 0.82 ABCB11 (0.57) ABCB11HRH1CCR3LMNAMEN1
Trifluoroacetic Acid SCHEMBL3150378 0.81 ABCB11 (0.57) ABCB11HRH1CCR3LMNAMEN1
SCHEMBL1682980 0.81 ABCB11 (0.74) ABCB11HRH1CCR3LMNAMEN1
SCHEMBL3048644 0.80 ABCB11 (0.60) ABCB11HRH1CCR3LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4115885-A1 A PHARMACEUTICAL COMPOSITION COMPRISING BAY 86-5277 AND SALTS THEREOF FOR USE IN THE TREATMENT OF VIRAL INFECTIONS AND HYPERINFLAMMATION Charité - Universitätsmedizin Berlin (DE) 2023-01-11 EP disclosed