SCHEMBL30176388

SCHEMBL30176388

Cc1cc(-n2c(C)c(C#N)c3cc(OCc4ccccc4)c(N=C(c4ccccc4)c4ccccc4)cc32)ccc1F

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 5/20 0.35
AS3MT Q9HBK9 1/20 0.35
PTGER1 P34995 6/20 0.34
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
TSHR P16473 1/20 0.33
HTT P42858 1/20 0.33
CYP2C9 P11712 1/20 0.33
KDM1A O60341 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23886672 1.00 MRGPRX4 (0.35) MRGPRX4AS3MTPTGER1LMNAMAPT
SCHEMBL23898683 0.83 AS3MT (0.38) AS3MTPTGER1LMNAMAPTTSHR
SCHEMBL30176398 0.83 AS3MT (0.42) AS3MTPTGER1LMNAMAPTTSHR
SCHEMBL23886810 0.83 AS3MT (0.42) AS3MTPTGER1LMNAMAPTTSHR
SCHEMBL23898684 0.71 AS3MT (0.40) AS3MTLMNAMAPTTSHRHTT
SCHEMBL23898401 0.69 KDM4E (0.35) LMNAMAPTTSHRHTT
SCHEMBL26652990 0.68 KDM4E (0.36) LMNAMAPTTSHRHTT
SCHEMBL30335469 0.67 PTGER1 (0.37) PTGER1MAPTKDM1A
SCHEMBL23883823 0.67 PTGER1 (0.37) PTGER1MAPTKDM1A
SCHEMBL23886911 0.67 LMNA (0.36) LMNAMAPTTSHRKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115916749-A Substituted 5-hydroxyindole compounds as alpha-1 antitrypsin modulators 弗特克斯药品有限公司 2023-04-04 CN disclosed
EP-4126817-A1 SUBSTITUTED 5-HYDROXYINDOLE COMPOUNDS AS MODULATORS OF ALPHA-1 ANTITRYPSIN Vertex Pharmaceuticals Incorporated (US) 2023-02-08 EP disclosed