SCHEMBL30179259

SCHEMBL30179259

CCOC(=O)N1CCCN(C2CCC3(CC2)CNc2ncccc23)CC1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.52
CHRM4 P08173 4/20 0.49
CHRM2 P08172 1/20 0.49
CHRM1 P11229 1/20 0.45
NOS2 P35228 1/20 0.44
MAPK1 P28482 1/20 0.41
GRIN2B Q13224 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20066060 1.00 KCNH2 (0.52) KCNH2CHRM4CHRM2CHRM1NOS2
SCHEMBL23778242 0.86 HRH3 (0.40)
SCHEMBL21120271 0.85 CHRM4 (0.47) KCNH2CHRM4CHRM2CHRM1NOS2
SCHEMBL30179252 0.85 KCNH2 (0.53) KCNH2CHRM4CHRM2CHRM1NOS2
SCHEMBL20066057 0.85 KCNH2 (0.53) KCNH2CHRM4CHRM2CHRM1NOS2
SCHEMBL30179198 0.81 KCNH2 (0.69) KCNH2CHRM4CHRM2CHRM1NOS2
SCHEMBL20066061 0.81 KCNH2 (0.69) KCNH2CHRM4CHRM2CHRM1NOS2
SCHEMBL23799176 0.80 KCNH2 (0.51) KCNH2CHRM4CHRM2CHRM1NOS2
SCHEMBL23799236 0.80 KDM4E (0.38) KCNH2GRIN2B
SCHEMBL20066064 0.79 CHRM4 (0.48) KCNH2CHRM4CHRM2CHRM1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109996792-B Heterocyclic compounds having activity as modulators of muscarinic M1 and/or M4 receptors in the treatment of CNS diseases and pain 赫普泰雅治疗有限公司 2023-02-17 CN disclosed