SCHEMBL30179252

SCHEMBL30179252

CCOC(=O)N1CCCN(C2CCC3(CC2)C(=O)Nc2ncccc23)CC1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 12/20 0.53
CHRM4 P08173 4/20 0.47
CHRM2 P08172 2/20 0.47
MAPK1 P28482 1/20 0.42
NOS2 P35228 1/20 0.42
CHRM1 P11229 2/20 0.42
CHRM5 P08912 1/20 0.40
CHRM3 P20309 1/20 0.40
CALCRL Q16602 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GRIN2B Q13224 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20066057 1.00 KCNH2 (0.53) KCNH2CHRM4CHRM2MAPK1NOS2
SCHEMBL23778441 0.87 CALCRL (0.40) CALCRLALDH1A1
SCHEMBL20066064 0.86 CHRM4 (0.48) KCNH2CHRM4CHRM2MAPK1NOS2
SCHEMBL20066060 0.85 KCNH2 (0.52) KCNH2CHRM4CHRM2MAPK1NOS2
SCHEMBL30179259 0.85 KCNH2 (0.52) KCNH2CHRM4CHRM2MAPK1NOS2
SCHEMBL30179395 0.85 OPRM1 (0.46) KCNH2CHRM4CHRM2MAPK1CHRM1
SCHEMBL20066046 0.85 OPRM1 (0.46) KCNH2CHRM4CHRM2MAPK1CHRM1
SCHEMBL30179222 0.84 MAPK1 (0.41) KCNH2CHRM4CHRM2MAPK1NOS2
SCHEMBL20066058 0.84 MAPK1 (0.41) KCNH2CHRM4CHRM2MAPK1NOS2
SCHEMBL21120271 0.84 CHRM4 (0.47) KCNH2CHRM4CHRM2MAPK1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109996792-B Heterocyclic compounds having activity as modulators of muscarinic M1 and/or M4 receptors in the treatment of CNS diseases and pain 赫普泰雅治疗有限公司 2023-02-17 CN disclosed