SCHEMBL30187948

SCHEMBL30187948

Nc1ncnc2c1sc1ncccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 11/20 1.00
LIMK1 P53667 8/20 1.00
CDC7 O00311 3/20 1.00
DBF4 Q9UBU7 2/20 1.00
CDK5 Q00535 2/20 0.61
CDK5R1 Q15078 1/20 0.61
KDM4E B2RXH2 1/20 0.59
NPC1 O15118 1/20 0.59
USP2 O75604 1/20 0.59
ALDH1A1 P00352 1/20 0.59
MAPT P10636 1/20 0.59
HPGD P15428 1/20 0.59
HSD17B10 Q99714 1/20 0.59
PIK3CA P42336 1/20 0.53
PLK4 O00444 1/20 0.53
AURKA O14965 1/20 0.53
DAPK3 O43293 1/20 0.53
DYRK3 O43781 1/20 0.53
ROCK2 O75116 1/20 0.53
PRKD3 O94806 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12807147 1.00 CLK1 (1.00) CLK1LIMK1CDC7DBF4CDK5
SCHEMBL16281249 0.80 CLK1 (0.67) CLK1LIMK1CDC7DBF4CDK5
SCHEMBL9042411 0.80 CLK1 (0.67) CLK1LIMK1CDC7DBF4CDK5
SCHEMBL30093319 0.80 CLK1 (0.67) CLK1LIMK1CDC7DBF4CDK5
SCHEMBL19738188 0.79 CLK1 (0.65) CLK1LIMK1CDC7DBF4CDK5
SCHEMBL30186939 0.79 CLK1 (0.65) CLK1LIMK1CDC7DBF4CDK5
SCHEMBL14115537 0.76 CLK1 (0.61) CLK1LIMK1CDC7DBF4KDM4E
SCHEMBL20609579 0.76 CLK1 (0.61) CLK1LIMK1CDC7DBF4CDK5
SCHEMBL14090789 0.76 CLK1 (0.61) CLK1LIMK1CDC7DBF4CDK5
SCHEMBL20120214 0.76 CLK1 (0.61) CLK1LIMK1CDC7DBF4CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116178391-A Forward allosteric modulators of muscarinic acetylcholine receptor M4 范德比尔特大学 2023-05-30 CN disclosed
CN-109310668-B Positive allosteric modulators of muscarinic acetylcholine receptor M4 范德比尔特大学 2023-01-24 CN disclosed