SCHEMBL30189809

SCHEMBL30189809

Cc1cc(Cl)nc2sc(Br)nc12

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.33
KDM4E B2RXH2 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C19 P33261 1/20 0.32
HIF1A Q16665 1/20 0.32
HSD17B10 Q99714 1/20 0.31
NQO2 P16083 1/20 0.30
ADORA3 P0DMS8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19783530 1.00 LMNA (0.33) LMNAKDM4ECYP3A4CYP2C19HIF1A
SCHEMBL28383665 0.82 GAA (0.35) LMNAKDM4ECYP3A4CYP2C19HIF1A
SCHEMBL19782603 0.79 HSD17B10 (0.49) LMNACYP3A4HSD17B10ADORA3
SCHEMBL30189823 0.79 HSD17B10 (0.49) LMNACYP3A4HSD17B10ADORA3
SCHEMBL30189475 0.74 RECQL (0.38) LMNAKDM4ENQO2
SCHEMBL19783074 0.74 RECQL (0.38) LMNAKDM4ENQO2
SCHEMBL25250290 0.73 AR (0.30)
SCHEMBL22392824 0.72 MAPT (0.40) KDM4EADORA3
SCHEMBL1129623 0.69 LMNA (0.44) LMNAKDM4ECYP3A4CYP2C19HIF1A
SCHEMBL22392806 0.68 BACE1 (0.51) LMNAKDM4EHSD17B10NQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed