Jnj-42165279

Jnj-42165279

SCHEMBL30201425

O=C(Nc1cnccc1Cl)N1CCN(Cc2ccc3c(c2)OC(F)(F)O3)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

FAAH

The experimentally established mechanism targets of Jnj-42165279. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FAAH known ✓ O00519 16/20 1.00
CYP2D6 P10635 2/20 1.00
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA9 Q16790 1/20 0.48
MAPK1 P28482 1/20 0.48
MCHR1 Q99705 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Jnj-42165279 SCHEMBL2585102 1.00 FAAH (1.00) FAAHCYP2D6CA12CA1CA2
Jnj-42165279 SCHEMBL29392521 1.00 FAAH (1.00) FAAHCYP2D6CA12CA1CA2
Jnj-42165279 SCHEMBL31616215 0.99 FAAH (0.98) FAAHCYP2D6CA12CA1CA2
Jnj-42165279 SCHEMBL2588988 0.99 FAAH (0.98) FAAHCYP2D6CA12CA1CA2
SCHEMBL15673544 0.86 FAAH (0.76) FAAHCYP2D6MCHR1
SCHEMBL3590970 0.84 FAAH (1.00) FAAHCYP2D6MAPK1
SCHEMBL2593197 0.83 FAAH (1.00) FAAHCYP2D6
SCHEMBL3637158 0.83 FAAH (0.76) FAAHCYP2D6MAPK1
SCHEMBL3598626 0.81 FAAH (1.00) FAAHCYP2D6MAPK1
SCHEMBL1277125 0.81 FAAH (0.68) FAAHCYP2D6MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115616216-A Use of an agent that inhibits or blocks the interaction between FAAH and NLRP3 华南理工大学 2023-01-17 CN claimed
WO-2025120480-A1 METHODS FOR TREATING SUBJECTS WITH AUTISM SPECTRUM DISORDER JANSSEN PHARMACEUTICA NV (BE) 2025-06-12 WO disclosed
WO-2024225481-A1 AGENT FOR IMPROVING THERAPEUTIC RESPONSIVENESS IN CANCER IMMUNOTHERAPY WITH PD-1 INHIBITOR OR PD-L1 INHIBITOR 国立大学法人京都大学 2024-10-31 WO disclosed
WO-2024102802-A1 ZELATRIAZIN FOR THE TREATMENT OF DEPRESSION TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2024-05-16 WO disclosed
CN-115616216-A Use of an agent that inhibits or blocks the interaction between FAAH and NLRP3 华南理工大学 2023-01-17 CN disclosed