SCHEMBL30212372

SCHEMBL30212372

c1ccc(OCc2ccnc(-n3ccnn3)n2)cc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.49
CYSLTR2 Q9NS75 1/20 0.43
CYSLTR1 Q9Y271 1/20 0.43
CYP19A1 P11511 3/20 0.40
NOTUM Q6P988 1/20 0.38
MAPT P10636 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
GRM5 P41594 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
FFAR1 O14842 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
PDE5A O76074 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24921074 0.81 CYP19A1 (0.39) CYP19A1NOTUM
SCHEMBL30212486 0.77 KCNH2 (0.47) KCNH2CYSLTR2CYSLTR1CYP19A1MAPT
SCHEMBL30212206 0.77 KCNH2 (0.54) KCNH2CYSLTR2CYSLTR1CYP19A1MAPT
SCHEMBL30212185 0.76 CYP19A1 (0.43) CYP19A1
SCHEMBL30212351 0.70 KCNH2 (0.43) KCNH2CYSLTR2CYSLTR1RAB9AGRM5
SCHEMBL1188120 0.70 CYP19A1 (0.60) CYP19A1NOTUMMAPTNPC1RAB9A
SCHEMBL17898216 0.69 KCNH2 (0.61) KCNH2CYSLTR2CYSLTR1CYP19A1MAPT
SCHEMBL20746692 0.69 KCNH2 (0.61) KCNH2CYSLTR2CYSLTR1MAPTNPC1
SCHEMBL28020279 0.67 NOTUM (0.44) CYP19A1NOTUM
SCHEMBL30212517 0.66 NPC1 (0.36) KCNH2CYP19A1MAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed