SCHEMBL30212751

SCHEMBL30212751

COc1cc(F)c(CO)nc1-c1c(C)cccc1C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
MAPT P10636 2/20 0.34
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34
G6PD P11413 1/20 0.34
PKM P14618 1/20 0.34
NQO2 P16083 1/20 0.34
PDCD1 Q15116 1/20 0.34
CD274 Q9NZQ7 1/20 0.34
ALDH1A1 P00352 2/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MAP4K1 Q92918 1/20 0.34
S1PR1 P21453 1/20 0.34
ADORA2A P29274 2/20 0.33
PDE4A P27815 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24028061 1.00 NPC1 (0.34) NPC1RAB9AMAPTLMNAPOLB
SCHEMBL24028074 0.88 RPS6KA2 (0.36) L3MBTL1MAP4K1PDE4APDE4BPDE4C
SCHEMBL30213035 0.88 RPS6KA2 (0.36) L3MBTL1MAP4K1PDE4APDE4BPDE4C
SCHEMBL24028393 0.87 PDE4A (0.34) MAPTL3MBTL1S1PR1PDE4APDE4B
SCHEMBL30212933 0.79 HSP90AA1 (0.39) NPC1RAB9AMAPTLMNAPOLB
SCHEMBL24028217 0.79 HSP90AA1 (0.39) NPC1RAB9AMAPTLMNAPOLB
SCHEMBL30212881 0.78 ALDH1A1 (0.39) RAB9ALMNAPOLBALDH1A1SMN1; SMN2
SCHEMBL24028387 0.78 ALDH1A1 (0.39) RAB9ALMNAPOLBALDH1A1SMN1; SMN2
SCHEMBL24028389 0.76 ALDH1A1 (0.33) NPC1RAB9AMAPTLMNAPOLB
SCHEMBL30212963 0.76 ALDH1A1 (0.33) NPC1RAB9AMAPTLMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4149928-A1 IMIDAZOLE 3-OXIDE DERIVATIVE BASED ACSS2 INHIBITORS AND METHODS OF USE THEREOF Metabomed Ltd (IL) 2023-03-22 EP disclosed
CN-115697974-A Imidazole 3-oxide derivative based ACSS2 inhibitors and methods of use thereof 美特波米德有限公司 2023-02-03 CN disclosed