SCHEMBL30226989

SCHEMBL30226989

C=CC(=O)Nc1ccc(B2OC(C)(C)C(C)(C)O2)cc1F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 7/20 0.47
CA2 P00918 7/20 0.47
CA9 Q16790 7/20 0.47
ROCK1 Q13464 1/20 0.42
HIF1A Q16665 3/20 0.39
LPL P06858 1/20 0.39
LIPG Q9Y5X9 1/20 0.39
ALDH1A1 P00352 1/20 0.38
CYP2C19 P33261 1/20 0.38
TGM2 P21980 1/20 0.37
P4HB P07237 1/20 0.36
PDGFRB P09619 2/20 0.36
KDR P35968 2/20 0.36
F2 P00734 1/20 0.36
F11 P03951 1/20 0.36
PRSS1 P07477 1/20 0.36
PRSS2 P07478 1/20 0.36
PRSS3 P35030 1/20 0.36
CA12 O43570 1/20 0.35
CA3 P07451 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16123326 0.90 PDGFRB (0.42) CA1CA2CA9ROCK1HIF1A
SCHEMBL24992096 0.90 CA1 (0.40) CA1CA2CA9ROCK1HIF1A
SCHEMBL5899542 0.84 CA1 (0.51) CA1CA2CA9ROCK1HIF1A
SCHEMBL30124283 0.84 CA1 (0.51) CA1CA2CA9ROCK1HIF1A
SCHEMBL2635766 0.84 CA1 (0.51) CA1CA2CA9ROCK1HIF1A
SCHEMBL16099915 0.83 HIF1A (0.45) CA1CA2CA9HIF1ALPL
SCHEMBL30380201 0.83 HIF1A (0.45) CA1CA2CA9HIF1ALPL
SCHEMBL31391204 0.83 CA1 (0.53) CA1CA2CA9ROCK1HIF1A
SCHEMBL21198519 0.82 GAA (0.41) HIF1AALDH1A1TGM2EGFRDGAT1
SCHEMBL31568575 0.82 CA1 (0.47) CA1CA2CA9ROCK1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023011581-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL APPLICATION THEREOF 江苏恒瑞医药股份有限公司 2023-02-09 WO disclosed