SCHEMBL30227253

SCHEMBL30227253

CCCCN1C(=O)[C@@H]([C@H](O)C2CCOCC2)NC(=O)C12CCN(Cc1ccc(Oc3ccc(NC(=O)C(C)C)cc3OC)cc1)CC2

nearest known ligand 0.63

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 20/20 0.63
CYP2C9 P11712 3/20 0.59
CYP2D6 P10635 2/20 0.59
CXCR4 P61073 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6186357 1.00 CCR5 (0.63) CCR5CYP2C9CYP2D6CXCR4
Hydrochloric Acid SCHEMBL5578702 0.99 CCR5 (0.63) CCR5CYP2C9CYP2D6CXCR4
Hydrochloric Acid SCHEMBL5578699 0.99 CCR5 (0.63) CCR5CYP2C9CYP2D6CXCR4
Hydrochloric Acid SCHEMBL6190007 0.93 CCR5 (0.65) CCR5CYP2C9CYP2D6CXCR4
SCHEMBL30227190 0.93 CCR5 (0.61) CCR5CYP2C9CYP2D6CXCR4
SCHEMBL6186771 0.93 CCR5 (0.61) CCR5CYP2C9CYP2D6CXCR4
Hydrochloric Acid SCHEMBL5578727 0.92 CCR5 (0.62) CCR5CYP2C9CYP2D6CXCR4
Hydrochloric Acid SCHEMBL5578730 0.92 CCR5 (0.62) CCR5CYP2C9CYP2D6CXCR4
SCHEMBL6186982 0.92 CCR5 (0.69) CCR5CYP2C9CYP2D6CXCR4
Hydrochloric Acid SCHEMBL6189902 0.91 CCR5 (0.70) CCR5CYP2C9CYP2D6CXCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4143235-A1 METHODS AND COMPOSITIONS FOR TREATING CYTOKINE STORM INFECTIONS, INCLUDING COVID-19, BY INHIBITING CCR5/CCL5 INTERACTION IncellDx, Inc. (US) 2023-03-08 EP disclosed