SCHEMBL30229307

SCHEMBL30229307

N#Cc1cnn2c1C(=O)NCC2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.36
PLAT P00750 2/20 0.34
CDC7 O00311 1/20 0.34
ALOX5 P09917 3/20 0.33
ALOX5AP P20292 3/20 0.33
FEN1 P39748 3/20 0.33
POLB P06746 1/20 0.33
HTT P42858 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CDK2 P24941 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
ABCB11 O95342 1/20 0.31
SLCO1B1 Q9Y6L6 1/20 0.31
P2RX7 Q99572 1/20 0.31
PTGS2 P35354 1/20 0.31
PKM P14618 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16402566 0.75 PARP1 (0.38) PARP1CDC7ALOX5ALOX5APFEN1
SCHEMBL16682624 0.75 CDC7 (0.36) PARP1PLATCDC7ALOX5ALOX5AP
SCHEMBL18209656 0.75 CDC7 (0.36) PARP1CDC7ALOX5ALOX5APFEN1
SCHEMBL18198141 0.75 PARP1 (0.38) PARP1CDC7ALOX5ALOX5APFEN1
Hydrochloric Acid SCHEMBL18209674 0.73 CDC7 (0.36) PARP1CDC7ALOX5ALOX5APFEN1
SCHEMBL20400002 0.73 CDC7 (0.33) PARP1CDC7ALOX5ALOX5APFEN1
SCHEMBL18215199 0.71 ALOX5 (0.41) PARP1CDC7ALOX5ALOX5APFEN1
SCHEMBL27199355 0.70 CYP1A2 (0.39) PARP1CDC7ALOX5ALOX5APFEN1
SCHEMBL26988582 0.70 ALOX5 (0.36) PARP1PLATCDC7ALOX5ALOX5AP
SCHEMBL16682636 0.69 PARP1 (0.45) PARP1PLATCDC7ALOX5ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3749669-B3 AHR MODULATORS IDEAYA BIOSCIENCES INC (US) 2024-09-04 EP claimed
EP-3749669-B1 AHR MODULATORS IDEAYA BIOSCIENCES INC (US) 2023-03-08 EP claimed