SCHEMBL30239369

SCHEMBL30239369

Cc1[nH]nc(-c2ccccc2)c1-c1ccc(-c2cnc3c(c2)CC(=O)N3)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 6/20 0.68
ABL1 P00519 2/20 0.68
CHEK1 O14757 1/20 0.68
AURKA O14965 1/20 0.68
DAPK3 O43293 1/20 0.68
PRKD3 O94806 1/20 0.68
MAP4K4 O95819 1/20 0.68
NTRK1 P04629 1/20 0.68
CSF1R P07333 1/20 0.68
RET P07949 1/20 0.68
MET P08581 1/20 0.68
PDGFRB P09619 1/20 0.68
PIM1 P11309 1/20 0.68
FGFR1 P11362 1/20 0.68
PDGFRA P16234 1/20 0.68
FLT1 P17948 1/20 0.68
LTK P29376 1/20 0.68
GRK5 P34947 1/20 0.68
KDR P35968 1/20 0.68
MAP2K2 P36507 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24963530 0.90 LRRK2 (0.53) LRRK2ABL1CHEK1AURKADAPK3
SCHEMBL5873863 0.83 KDR (1.00) LRRK2ABL1CHEK1AURKADAPK3
SCHEMBL11192094 0.74 AKT2 (0.68) LRRK2CHEK1CNR1CNR2GPR55
SCHEMBL13854137 0.73 ABL1 (0.74) LRRK2ABL1CHEK1AURKADAPK3
SCHEMBL13854158 0.71 ABL1 (0.67) LRRK2ABL1CHEK1AURKADAPK3
SCHEMBL3141083 0.71 ABL1 (0.76) LRRK2ABL1CHEK1AURKADAPK3
SCHEMBL23524008 0.71 ABL1 (0.66) LRRK2ABL1CHEK1AURKADAPK3
SCHEMBL30239363 0.71 PDE3B (0.56) LRRK2
SCHEMBL24964988 0.69 IKBKB (0.58) LRRK2CHEK1IKBKECNR1CNR2
SCHEMBL1396298 0.69 ABL1 (0.67) LRRK2ABL1CHEK1AURKADAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023004280-A1 SELECTIVE PYRAZOLE LRRK2 INHIBITORS AND METHODS FOR USE THEREOF THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2023-01-26 WO claimed