SCHEMBL3024265

SCHEMBL3024265

Cc1c(N[C@H]2CC[C@H](N)CC2)nn2ccnc2c1Nc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 3/20 0.48
CDK2 P24941 7/20 0.44
FLT3 P36888 5/20 0.44
CCNE1 P24864 5/20 0.44
MAPKAPK2 P49137 7/20 0.43
PDGFRA P16234 4/20 0.42
SRC P12931 1/20 0.42
ADORA3 P0DMS8 2/20 0.37
ADORA2A P29274 2/20 0.37
ADORA1 P30542 2/20 0.37
MAPK9 P45984 1/20 0.37
MAPK10 P53779 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3021965 0.91 ADORA3 (0.43) MAPK8CDK2FLT3CCNE1MAPKAPK2
SCHEMBL3026215 0.91 ADORA3 (0.43) MAPK8CDK2FLT3CCNE1MAPKAPK2
SCHEMBL3021971 0.91 ADORA3 (0.43) MAPK8CDK2FLT3CCNE1MAPKAPK2
SCHEMBL3015203 0.91 MAPKAPK2 (0.47) MAPK8CDK2FLT3CCNE1MAPKAPK2
SCHEMBL3020113 0.89 FLT3 (0.42) MAPK8CDK2FLT3CCNE1MAPKAPK2
SCHEMBL3020115 0.89 FLT3 (0.42) MAPK8CDK2FLT3CCNE1MAPKAPK2
SCHEMBL3025252 0.89 CDK2 (0.47) MAPK8CDK2FLT3CCNE1MAPKAPK2
SCHEMBL3025258 0.89 CDK2 (0.47) MAPK8CDK2FLT3CCNE1MAPKAPK2
SCHEMBL3022048 0.88 FLT3 (0.45) MAPK8CDK2FLT3CCNE1MAPKAPK2
SCHEMBL3022042 0.88 FLT3 (0.45) MAPK8CDK2FLT3CCNE1MAPKAPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100204212-A1 FUSED HETEROCYCLIC COMPOUNDS USEFUL AS KINASE MODULATORS BRISTOL-MYERS SQUIBB COMPANY 2010-08-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100204212-A1 FUSED HETEROCYCLIC COMPOUNDS USEFUL AS KINASE MODULATORS MAP2K2, MAP3K2, MAP4K2 MAPK8 84/4885CDK2 40/4885FLT3 345/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.