SCHEMBL302427

SCHEMBL302427

CCc1ccc(S(=O)(=O)N(Cc2ccccc2)c2ccc(C(=O)N3CCN(c4ccccc4)CC3)cc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.68
HPGD P15428 2/20 0.68
LMNA P02545 5/20 0.67
SMN1; SMN2 Q16637 3/20 0.62
HTT P42858 2/20 0.62
GAA P10253 2/20 0.56
CNR2 P34972 3/20 0.54
CA12 O43570 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA7 P43166 1/20 0.54
CA9 Q16790 1/20 0.54
CA14 Q9ULX7 1/20 0.54
RAB9A P51151 1/20 0.53
PTGES O14684 2/20 0.52
ALOX5 P09917 2/20 0.52
CNR1 P21554 1/20 0.52
MEN1 O00255 3/20 0.51
MAPK1 P28482 1/20 0.51
MAPT P10636 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL303307 0.92 LMNA (0.71) KMT2AHPGDLMNASMN1; SMN2HTT
SCHEMBL303907 0.91 LMNA (0.65) KMT2AHPGDLMNASMN1; SMN2HTT
SCHEMBL302243 0.89 LMNA (0.62) KMT2AHPGDLMNASMN1; SMN2HTT
SCHEMBL1711093 0.89 LMNA (0.71) KMT2AHPGDLMNASMN1; SMN2HTT
SCHEMBL302271 0.87 LMNA (0.68) KMT2AHPGDLMNASMN1; SMN2HTT
SCHEMBL3282269 0.87 LMNA (0.68) KMT2AHPGDLMNASMN1; SMN2HTT
SCHEMBL303534 0.87 KMT2A (0.61) KMT2AHPGDLMNASMN1; SMN2HTT
SCHEMBL1711088 0.87 LMNA (0.59) KMT2AHPGDLMNASMN1; SMN2HTT
SCHEMBL1723106 0.85 HTR2C (0.63) KMT2AHPGDLMNASMN1; SMN2HTT
SCHEMBL13065013 0.85 CNR2 (0.61) KMT2AHPGDLMNASMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2344456-B1 NOVEL POTASSIUM CHANNEL BLOCKER JAPAN TOBACCO INC (JP) 2018-07-25 EP claimed
US-8258138-B2 Potassium channel blockers XENTION LIMITED (GB) 2012-09-04 US claimed
JP-2012500834-A 2012-01-12 JP claimed
EP-2344456-A1 NOVEL POTASSIUM CHANNEL BLOCKER Xention Limited (GB) 2011-07-20 EP claimed
US-20100087437-A1 Novel Potassium Channel Blockers XENTION LIMITED (GB) 2010-04-08 US claimed
WO-2010023445-A1 NOVEL POTASSIUM CHANNEL BLOCKER XENTION LIMITED (GB) 2010-03-04 WO claimed
EP-2344456-B1 NOVEL POTASSIUM CHANNEL BLOCKER JAPAN TOBACCO INC (JP) 2018-07-25 EP disclosed
US-8258138-B2 Potassium channel blockers XENTION LIMITED (GB) 2012-09-04 US disclosed
US-20100087437-A1 Novel Potassium Channel Blockers XENTION LIMITED (GB) 2010-04-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100087437-A1 Novel Potassium Channel Blockers KCNB1, KCNJ2, KCNJ11 KMT2A 777/4885HPGD 3739/4885LMNA 1683/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.