SCHEMBL30252544

SCHEMBL30252544

Nc1cc(-c2nccs2)nc(-c2ccccn2)c1Br

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 8/20 0.43
HSP90AA1 P07900 1/20 0.42
RAB9A P51151 1/20 0.40
PDPK1 O15530 1/20 0.37
ADORA1 P30542 7/20 0.37
KDM4E B2RXH2 2/20 0.37
NPC1 O15118 1/20 0.37
HDAC2 Q92769 1/20 0.36
SYK P43405 1/20 0.36
ALOX15 P16050 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CYP19A1 P11511 1/20 0.35
PDE10A Q9Y233 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30252710 0.86 ADORA2A (0.42) ADORA2AHSP90AA1RAB9APDPK1ADORA1
SCHEMBL20911213 0.86 ADORA2A (0.42) ADORA2AHSP90AA1RAB9APDPK1ADORA1
SCHEMBL30252375 0.84 ADORA2A (0.58) ADORA2AHSP90AA1RAB9AADORA1SYK
SCHEMBL20911255 0.84 ADORA2A (0.58) ADORA2AHSP90AA1RAB9AADORA1SYK
SCHEMBL30252574 0.84 ADORA2A (0.40) ADORA2AHSP90AA1RAB9APDPK1ADORA1
SCHEMBL20911240 0.83 CCR1 (0.47) ADORA2AHSP90AA1RAB9AADORA1KDM4E
SCHEMBL30252590 0.82 HSP90AA1 (0.43) ADORA2AHSP90AA1RAB9AADORA1SYK
SCHEMBL20911188 0.81 KDM4E (0.47) ADORA2AHSP90AA1RAB9APDPK1ADORA1
SCHEMBL30252648 0.81 ADORA2A (0.40) ADORA2AHSP90AA1RAB9AADORA1SYK
SCHEMBL20911562 0.77 ADORA2A (0.41) ADORA2AHSP90AA1RAB9AADORA1SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109651358-B 4-aminopyridine derivative, pharmaceutical composition, preparation method and application thereof 上海迪诺医药科技有限公司 2023-04-07 CN disclosed