SCHEMBL30252574

SCHEMBL30252574

Nc1cc(-c2nccs2)nc(-c2cccc(F)n2)c1Br

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.40
HSP90AA1 P07900 1/20 0.40
CYP1A1 P04798 4/20 0.38
CYP1A2 P05177 4/20 0.38
CYP1B1 Q16678 4/20 0.38
RAB9A P51151 1/20 0.35
ADK P55263 1/20 0.35
ADORA1 P30542 3/20 0.34
SYK P43405 3/20 0.33
SRC P12931 1/20 0.33
CDK2 P24941 1/20 0.33
ZAP70 P43403 1/20 0.33
LOXL2 Q9Y4K0 1/20 0.32
PDPK1 O15530 1/20 0.32
HPGD P15428 1/20 0.32
CFTR P13569 1/20 0.32
PIM1 P11309 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30252710 0.88 ADORA2A (0.42) ADORA2AHSP90AA1CYP1A1CYP1A2CYP1B1
SCHEMBL20911213 0.88 ADORA2A (0.42) ADORA2AHSP90AA1CYP1A1CYP1A2CYP1B1
SCHEMBL30252544 0.84 ADORA2A (0.43) ADORA2AHSP90AA1RAB9AADORA1SYK
SCHEMBL30252590 0.81 HSP90AA1 (0.43) ADORA2AHSP90AA1CYP1A1CYP1A2CYP1B1
SCHEMBL20911255 0.81 ADORA2A (0.58) ADORA2AHSP90AA1CYP1A1CYP1A2CYP1B1
SCHEMBL30252375 0.81 ADORA2A (0.58) ADORA2AHSP90AA1CYP1A1CYP1A2CYP1B1
SCHEMBL30252750 0.80 SYK (0.38) ADORA2AHSP90AA1SYKSRCCDK2
SCHEMBL20911562 0.79 ADORA2A (0.41) ADORA2AHSP90AA1CYP1A1CYP1A2CYP1B1
SCHEMBL30252564 0.79 ADORA2A (0.41) ADORA2AHSP90AA1CYP1A1CYP1A2CYP1B1
SCHEMBL20911608 0.76 MAP4K4 (0.38) ADORA2AADORA1PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109651358-B 4-aminopyridine derivative, pharmaceutical composition, preparation method and application thereof 上海迪诺医药科技有限公司 2023-04-07 CN disclosed