SCHEMBL30253333

SCHEMBL30253333

NC1(C(=O)O)Cc2cccc(Cl)c2C1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 2/20 0.41
GRM3 Q14832 1/20 0.41
AKR1B1 P15121 1/20 0.38
ADRA2A P08913 3/20 0.37
ADRA2B P18089 2/20 0.37
ADRA2C P18825 2/20 0.37
ADRA1D P25100 2/20 0.37
ADRA1A P35348 2/20 0.37
ADRA1B P35368 2/20 0.37
TAAR1 Q96RJ0 1/20 0.37
HDAC11 Q96DB2 1/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
CYP1A2 P05177 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
HSD17B10 Q99714 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23857362 1.00 GRM2 (0.41) GRM2GRM3AKR1B1ADRA2AADRA2B
SCHEMBL4599994 0.86 GRM2 (0.39) GRM2GRM3AKR1B1ADRA2AADRA2B
SCHEMBL8828732 0.86 ADRA2A (0.46) GRM2GRM3AKR1B1ADRA2AADRA2B
SCHEMBL23857218 0.81 HDAC11 (0.36) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL27775131 0.80 HTR2A (0.35) GRM2GRM3ADRA2AADRA2BADRA2C
SCHEMBL3304544 0.78 BRD4 (0.40) ADRA1AKDM4EALDH1A1CYP1A2TSHR
SCHEMBL29476532 0.78 HDAC9 (0.44) GRM2
SCHEMBL122942 0.78 HDAC9 (0.44) GRM2
SCHEMBL23857123 0.76 AKR1B1 (0.42) GRM2GRM3AKR1B1ADRA2AADRA2B
SCHEMBL8649961 0.76 ADRA2A (0.46) ADRA2AADRA2BADRA2CADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4126855-A1 COMPOUNDS AND THEIR USE IN THE TREATMENT OF BACTERIAL INFECTION F. Hoffmann-La Roche AG (CH) 2023-02-08 EP disclosed