SCHEMBL3025664

SCHEMBL3025664

CC(N)c1ccc(B2OC(C)(C)C(C)(C)O2)cc1Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.50
TP53 P04637 1/20 0.50
HTT P42858 1/20 0.50
LPL P06858 11/20 0.40
LIPG Q9Y5X9 11/20 0.40
AAK1 Q2M2I8 1/20 0.39
CA1 P00915 3/20 0.38
CA2 P00918 3/20 0.38
CA9 Q16790 3/20 0.38
CA12 O43570 1/20 0.38
CA3 P07451 1/20 0.38
CA4 P22748 1/20 0.38
CA6 P23280 1/20 0.38
CA5A P35218 1/20 0.38
CA7 P43166 1/20 0.38
CA14 Q9ULX7 1/20 0.38
CA5B Q9Y2D0 1/20 0.38
F11 P03951 1/20 0.37
EGFR P00533 1/20 0.36
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25267227 0.86 LPL (0.41) LMNATP53HTTLPLLIPG
SCHEMBL25207380 0.86 LPL (0.41) LMNATP53HTTLPLLIPG
Hydrochloric Acid SCHEMBL25260965 0.84 LPL (0.40) LMNATP53HTTLPLLIPG
SCHEMBL9910113 0.84 PDE2A (0.44) LPLLIPGAAK1CA1CA2
SCHEMBL2699826 0.84 PDE2A (0.44) LPLLIPGAAK1CA1CA2
Hydrochloric Acid SCHEMBL25260963 0.84 LPL (0.40) LMNATP53HTTLPLLIPG
SCHEMBL2411421 0.83 LPL (0.44) LPLLIPGAAK1CA1CA2
SCHEMBL14758481 0.82 AAK1 (0.40) LPLLIPGAAK1CA1CA2
SCHEMBL31294725 0.81 LPL (0.46) LPLLIPGCA1CA2CA9
SCHEMBL4578027 0.80 AAK1 (0.39) LPLLIPGAAK1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2396301-A2 SMALL MOLECULE BRADYKININ B1 RECEPTOR ANTAGONISTS Jerini AG (DE) 2011-12-21 EP disclosed
WO-2010091876-A2 SMALL MOLECULE BRADYKININ B1 RECEPTOR ANTAGONISTS JERINI AG (DE) 2010-08-19 WO disclosed