SCHEMBL30257538

SCHEMBL30257538

Cn1nc(-c2nccs2)cc1Oc1cc(C#N)ccc1-c1ncc(CN)cn1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 7/20 0.35
NSD2 O96028 4/20 0.33
SCN9A Q15858 4/20 0.33
LOXL2 Q9Y4K0 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
SLC2A1 P11166 1/20 0.32
SLC2A3 P11169 1/20 0.32
SLC2A4 P14672 1/20 0.32
CYP19A1 P11511 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25554854 1.00 CRHR1 (0.35) CRHR1NSD2SCN9ALOXL2ADORA2A
SCHEMBL30257220 0.93 CRHR1 (0.34) CRHR1SCN9AADORA2AADORA1SLC2A1
SCHEMBL25554461 0.93 CRHR1 (0.34) CRHR1SCN9AADORA2AADORA1SLC2A1
SCHEMBL25554810 0.88 CRHR1 (0.33) CRHR1SCN9AADORA2AADORA1SLC2A1
SCHEMBL25555463 0.86 NSD2 (0.33) NSD2SCN9ACYP19A1CYP11B1CYP11B2
SCHEMBL25555468 0.86 NSD2 (0.33) NSD2SCN9A
SCHEMBL25555465 0.86 NSD2 (0.33) NSD2SCN9A
SCHEMBL30256868 0.85 CRHR1 (0.33) CRHR1NSD2SCN9ASLC2A1SLC2A3
SCHEMBL25554458 0.85 CRHR1 (0.33) CRHR1NSD2SCN9ASLC2A1SLC2A3
SCHEMBL25057937 0.85 GRM5 (0.37) NSD2CYP19A1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115996910-A Aryl or heteroaryl derivatives 帝人制药株式会社 2023-04-21 CN claimed
CN-115996910-A Aryl or heteroaryl derivatives 帝人制药株式会社 2023-04-21 CN disclosed
EP-4137481-A1 ARYL OR HETEROARYL DERIVATIVE Teijin Pharma Limited (JP) 2023-02-22 EP disclosed