SCHEMBL30258337

SCHEMBL30258337

COC(=O)c1nn(C)c2cc(Br)ccc12

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ELANE P08246 10/20 0.54
PLAU P00749 4/20 0.45
F2 P00734 3/20 0.45
PDGFRA P16234 1/20 0.43
CDK5 Q00535 1/20 0.43
TYRO3 Q06418 1/20 0.43
KDM4E B2RXH2 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.41
IRAK4 Q9NWZ3 1/20 0.41
HTR3A P46098 1/20 0.41
NR4A2 P43354 1/20 0.40
CTRB1 P17538 1/20 0.40
TSHR P16473 2/20 0.39
HTT P42858 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL498049 1.00 ELANE (0.54) ELANEPLAUF2PDGFRACDK5
SCHEMBL17419175 0.88 ELANE (0.64) ELANEPLAUF2KDM4EL3MBTL1
SCHEMBL31646748 0.88 ELANE (0.64) ELANEPLAUF2KDM4EL3MBTL1
SCHEMBL9959858 0.85 ELANE (0.57) ELANEPLAUF2MAPT
SCHEMBL492125 0.83 PDGFRA (0.47) ELANEPDGFRACDK5TYRO3KDM4E
SCHEMBL19128015 0.82 ELANE (0.45) ELANEPLAUF2KDM4EL3MBTL1
SCHEMBL498197 0.82 ELANE (0.51) ELANEPLAUF2PDGFRACDK5
SCHEMBL14011218 0.81 ELANE (0.44) ELANEPLAUF2KDM4EHTR3A
SCHEMBL19127362 0.81 ELANE (0.50) ELANEPLAUF2PDGFRACDK5
SCHEMBL22031821 0.80 ALDH1A1 (0.44) ELANEPLAUF2KDM4EHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4735452-A2 HETEROBIFUNCTIONAL COMPOUNDS FOR THE DEGRADATION OF KRAS PROTEIN Merck Patent GmbH (DE) 2026-05-06 EP disclosed
EP-4735438-A2 HETEROBIFUNCTIONAL COMPOUNDS FOR THE DEGRADATION OF KRAS Merck Patent GmbH (DE) 2026-05-06 EP disclosed
WO-2025006783-A2 HETEROBIFUNCTIONAL COMPOUNDS FOR THE DEGRADATION OF KRAS MERCK PATENT GMBH (DE) 2025-01-02 WO disclosed
WO-2025006753-A2 HETEROBIFUNCTIONAL COMPOUNDS FOR THE DEGRADATION OF KRAS PROTEIN MERCK PATENT GMBH (DE) 2025-01-02 WO disclosed
WO-2023059792-A1 CORONAVIRUS NON-STRUCTURAL PROTEIN 3 DEGRADING COMPOUNDS C4 THRAPEUTICS, INC. (US) 2023-04-13 WO disclosed