SCHEMBL30265752

SCHEMBL30265752

CC(C)N(C)C(=O)c1cc(F)ccc1-n1c(=S)n(C2CCCN(Cc3ccc4[nH]c(=O)[nH]c4c3)C2)c2ccncc21

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.34
TDO2 P48775 2/20 0.34
KDM4E B2RXH2 5/20 0.32
HTT P42858 1/20 0.32
LMNA P02545 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GRM2 Q14416 1/20 0.32
CYP3A4 P08684 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
MPO P05164 1/20 0.31
ALDH1A1 P00352 2/20 0.31
HPGD P15428 1/20 0.31
PKM P14618 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19972562 1.00 IDO1 (0.34) IDO1TDO2KDM4EHTTLMNA
SCHEMBL19972520 0.87 CYP3A4 (0.40) CYP3A4
SCHEMBL31001184 0.87 CYP3A4 (0.40) CYP3A4
SCHEMBL31001181 0.83 IDO1 (0.34) IDO1TDO2KDM4EHTTLMNA
SCHEMBL19972575 0.83 IDO1 (0.34) IDO1TDO2KDM4EHTTLMNA
SCHEMBL27197445 0.82 IDO1 (0.34) IDO1TDO2KDM4EHTTLMNA
SCHEMBL30266044 0.82 IDO1 (0.34) IDO1TDO2KDM4EHTTLMNA
SCHEMBL19972522 0.82 IDO1 (0.34) IDO1TDO2KDM4EHTTLMNA
SCHEMBL26006977 0.80 IDO1 (0.33) IDO1TDO2KDM4EHTTLMNA
SCHEMBL19972638 0.79 CDK9 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3512850-B1 INHIBITORS OF THE MENIN-MLL INTERACTION VITAE PHARMACEUTICALS LLC (US) 2023-04-12 EP claimed