SCHEMBL30272016

SCHEMBL30272016

ClCCCOc1cccc(Br)c1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 1/20 0.47
RAB9A P51151 6/20 0.41
NPC1 O15118 5/20 0.41
SMN1; SMN2 Q16637 4/20 0.41
CYP1A2 P05177 3/20 0.41
CYP2C19 P33261 3/20 0.41
TDP1 Q9NUW8 3/20 0.41
CYP3A4 P08684 2/20 0.41
TP53 P04637 1/20 0.41
CYP2D6 P10635 1/20 0.41
TSHR P16473 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HTR7 P34969 1/20 0.41
LMNA P02545 3/20 0.39
MAPT P10636 6/20 0.37
HPGD P15428 4/20 0.37
L3MBTL1 Q9Y468 4/20 0.37
KDM4E B2RXH2 3/20 0.37
CYP2C9 P11712 2/20 0.37
MAPK1 P28482 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18728740 1.00 MRGPRX4 (0.47) MRGPRX4RAB9ANPC1SMN1; SMN2CYP1A2
SCHEMBL30272015 1.00 MRGPRX4 (0.47) MRGPRX4RAB9ANPC1SMN1; SMN2CYP1A2
SCHEMBL28912849 0.94 MRGPRX4 (0.49) MRGPRX4RAB9ANPC1SMN1; SMN2CYP1A2
SCHEMBL28912859 0.92 MRGPRX4 (0.47) MRGPRX4RAB9ANPC1SMN1; SMN2CYP1A2
SCHEMBL18728495 0.87 MRGPRX4 (0.46) MRGPRX4RAB9ANPC1SMN1; SMN2CYP1A2
SCHEMBL29772011 0.87 MRGPRX4 (0.46) MRGPRX4RAB9ANPC1SMN1; SMN2CYP1A2
SCHEMBL11097966 0.86 CYP1A2 (0.47) RAB9ANPC1SMN1; SMN2CYP1A2CYP2C19
SCHEMBL18727941 0.85 HTR1B (0.50) MRGPRX4RAB9ANPC1SMN1; SMN2CYP1A2
SCHEMBL18704479 0.83 MRGPRX4 (0.46) MRGPRX4RAB9ANPC1SMN1; SMN2CYP1A2
SCHEMBL5661298 0.82 HTR7 (0.58) RAB9ANPC1SMN1; SMN2CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115466251-B Condensed heterocyclic compound, preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2024-06-21 CN disclosed
CN-109863146-B Biaryl compounds as immunomodulators 百时美施贵宝公司 2023-02-28 CN disclosed
CN-115466251-A Fused heterocyclic compound, preparation method thereof, pharmaceutical composition and application 中国医学科学院药物研究所 2022-12-13 CN disclosed