Pf-05241328

Pf-05241328

SCHEMBL30275387

Cc1nn(-c2cnc(OCC(C)C)c(Cl)c2)c2ccc(C(=O)NS(C)(=O)=O)cc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 20/20 1.00
SCN5A Q14524 12/20 0.61
CYP2C9 P11712 2/20 0.60
CYP2C8 P10632 1/20 0.60
CYP2B6 P20813 1/20 0.60
CYP2C19 P33261 1/20 0.60
SCN4A P35499 1/20 0.60
SCN2A Q99250 1/20 0.60
CYP3A4 P08684 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pf-05241328 SCHEMBL10324699 1.00 SCN9A (1.00) SCN9ASCN5ACYP2C9CYP2C8CYP2B6
SCHEMBL22484359 0.91 SCN9A (0.83) SCN9ASCN5ACYP2C9CYP2C8CYP2B6
SCHEMBL10378866 0.91 SCN9A (0.83) SCN9ASCN5ACYP2C9CYP2C8CYP2B6
SCHEMBL10379156 0.91 SCN9A (0.83) SCN9ASCN5ACYP2C9CYP2C8CYP2B6
SCHEMBL10380265 0.90 SCN9A (0.82) SCN9ASCN5ACYP2C9CYP2C8CYP2B6
SCHEMBL10380388 0.90 SCN9A (0.81) SCN9ASCN5ACYP2C9CYP2C8CYP2B6
SCHEMBL10380147 0.89 SCN9A (0.81) SCN9ASCN5ACYP2C9CYP2C8CYP2B6
SCHEMBL10326013 0.88 SCN9A (0.79) SCN9ASCN5ACYP2C9CYP2C8CYP2B6
SCHEMBL10379494 0.88 SCN9A (0.79) SCN9ASCN5A
SCHEMBL10379941 0.86 SCN9A (0.76) SCN9ASCN5ACYP2C9CYP2C8CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025106656-A1 METHODS OF PREVENTING OR REDUCING CARTILAGE LOSS AND/OR JOINT DAMAGE USING NAV 1.7 INHIBITORS YALE UNIVERSITY (US) 2025-05-22 WO claimed
WO-2025106656-A1 METHODS OF PREVENTING OR REDUCING CARTILAGE LOSS AND/OR JOINT DAMAGE USING NAV 1.7 INHIBITORS YALE UNIVERSITY (US) 2025-05-22 WO disclosed
CN-111285825-B Benzene sulfonamide substituted derivative, preparation method and application thereof 中国科学院上海药物研究所 2023-02-17 CN disclosed