SCHEMBL30280660

SCHEMBL30280660

N#Cc1ccnc(-c2ccsc2)c1C#N

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.48
ADORA1 P30542 3/20 0.48
ADORA2A P29274 2/20 0.48
CDK5 Q00535 1/20 0.41
CDK5R1 Q15078 1/20 0.41
TDO2 P48775 1/20 0.40
FLT4 P35916 1/20 0.40
MAPK8 P45983 1/20 0.40
MAPK9 P45984 1/20 0.40
CSNK2A1 P68400 1/20 0.40
DYRK1A Q13627 1/20 0.40
AURKB Q96GD4 1/20 0.40
PRKD2 Q9BZL6 1/20 0.40
PDE3A Q14432 1/20 0.36
RET P07949 4/20 0.34
CYP2A6 P11509 3/20 0.34
CYP2B6 P20813 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28954919 1.00 LRRK2 (0.48) LRRK2ADORA1ADORA2ACDK5CDK5R1
SCHEMBL3287223 0.79 LRRK2 (0.46) LRRK2ADORA1ADORA2ACDK5CDK5R1
SCHEMBL9359308 0.70 LRRK2 (0.43) LRRK2ADORA1ADORA2ATDO2PDE3A
SCHEMBL1028589 0.70 KDM1A (0.45) LRRK2ADORA1ADORA2AFLT4MAPK8
SCHEMBL11937878 0.69 LRRK2 (0.46) LRRK2ADORA1ADORA2ACDK5CDK5R1
SCHEMBL9680772 0.68 ADORA1 (0.55) ADORA1ADORA2ACDK5CDK5R1TDO2
SCHEMBL12470406 0.67 KDM4E (0.43) CDK5CDK5R1DYRK1AKDM4EMEN1
SCHEMBL1996285 0.65 LRRK2 (0.34) LRRK2CYP2C9CYP2C19KDM4EMEN1
SCHEMBL30701246 0.65 LRRK2 (0.34) LRRK2CYP2C9CYP2C19KDM4EMEN1
SCHEMBL16177867 0.65 LRRK2 (1.00) LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115710219-B Method for preparing meta-cyano-substituted pyridine compound 南开大学 2024-12-03 CN disclosed
CN-115710219-A Method for preparing meta cyano-substituted pyridine compound 南开大学 2023-02-24 CN disclosed