SCHEMBL30286355

SCHEMBL30286355

C[C@@H]1CN(c2ccc(C#N)cn2)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.58
HDAC1 Q13547 1/20 0.58
CHRM4 P08173 1/20 0.53
CHRM1 P11229 1/20 0.51
PARP1 P09874 5/20 0.51
PARP2 Q9UGN5 3/20 0.51
GPR119 Q8TDV5 3/20 0.48
PANK3 Q9H999 4/20 0.47
PDK1 Q15118 1/20 0.46
PDK2 Q15119 1/20 0.46
PIK3CD O00329 1/20 0.44
CHRM2 P08172 1/20 0.44
GRM1 Q13255 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26125207 1.00 MAP4K4 (0.58) MAP4K4HDAC1CHRM4CHRM1PARP1
SCHEMBL26128841 1.00 MAP4K4 (0.58) MAP4K4HDAC1CHRM4CHRM1PARP1
SCHEMBL30546539 1.00 MAP4K4 (0.58) MAP4K4HDAC1CHRM4CHRM1PARP1
SCHEMBL21522485 0.87 PARP1 (0.52) MAP4K4HDAC1CHRM4CHRM1PARP1
SCHEMBL24963042 0.86 GPR119 (0.58) MAP4K4HDAC1CHRM4CHRM1GPR119
SCHEMBL24963653 0.86 GPR119 (0.58) MAP4K4HDAC1CHRM4CHRM1GPR119
SCHEMBL26125148 0.84 PARP1 (0.58) CHRM4CHRM1PARP1PARP2PANK3
SCHEMBL28982891 0.84 PARP1 (0.58) CHRM4CHRM1PARP1PARP2PANK3
SCHEMBL23560717 0.84 MAP4K4 (0.52) MAP4K4HDAC1CHRM4GPR119PIK3CD
SCHEMBL23561132 0.84 MAP4K4 (0.52) MAP4K4HDAC1CHRM4GPR119PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4338737-A1 PARP7 INHIBITOR AND USE THEREOF Novostar Pharmaceuticals, Ltd. (CN) 2024-03-20 EP disclosed
CN-115785074-A PARP7 inhibitors and uses thereof 诺沃斯达药业(上海)有限公司 2023-03-14 CN disclosed