SCHEMBL30286390

SCHEMBL30286390

COC(=O)c1cc2[nH]ncc2cc1Br

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AXL P30530 1/20 0.56
MAPT P10636 2/20 0.50
TSHR P16473 1/20 0.47
NPC1 O15118 4/20 0.44
RAB9A P51151 4/20 0.44
NOS1 P29475 2/20 0.44
METAP2 P50579 2/20 0.44
DYRK1A Q13627 1/20 0.44
KDM4E B2RXH2 2/20 0.43
LMNA P02545 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ROCK2 O75116 2/20 0.42
ROCK1 Q13464 2/20 0.42
CASP6 P55212 1/20 0.42
ALDH1A1 P00352 2/20 0.41
CSNK2A1 P68400 1/20 0.40
MKNK1 Q9BUB5 1/20 0.40
MAOB P27338 2/20 0.39
POLB P06746 1/20 0.39
F2 P00734 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18554980 1.00 AXL (0.56) AXLMAPTTSHRNPC1RAB9A
SCHEMBL31602581 0.94 AXL (0.53) AXLMAPTTSHRNPC1RAB9A
SCHEMBL18183739 0.83 TSHR (0.49) AXLMAPTTSHRNPC1RAB9A
SCHEMBL617024 0.83 AXL (0.53) AXLMAPTNPC1RAB9ANOS1
SCHEMBL31041189 0.82 TSHR (0.55) AXLMAPTTSHRNPC1RAB9A
SCHEMBL1273838 0.82 TSHR (0.55) AXLMAPTTSHRNPC1RAB9A
SCHEMBL15687581 0.82 TSHR (0.47) AXLMAPTTSHRNPC1RAB9A
SCHEMBL30584955 0.82 TSHR (0.47) AXLMAPTTSHRNPC1RAB9A
SCHEMBL22446005 0.81 TSHR (0.50) AXLMAPTTSHRNPC1RAB9A
SCHEMBL22446038 0.81 CASP6 (0.54) AXLMAPTNPC1RAB9ANOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115873007-A Condensed tetracyclic derivative, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2023-03-31 CN disclosed