SCHEMBL30289809

SCHEMBL30289809

CC/C(=C(\c1ccccc1)c1ccc(Oc2ccccc2OC(C)N(C)C)cc1)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 10/20 0.52
ESR2 Q92731 6/20 0.52
MAPT P10636 3/20 0.52
CYP3A4 P08684 3/20 0.52
MEN1 O00255 2/20 0.52
TP53 P04637 2/20 0.52
PGR P06401 2/20 0.52
ESRRG P62508 2/20 0.52
KMT2A Q03164 2/20 0.52
NPC1 O15118 1/20 0.52
NR1I2 O75469 1/20 0.52
PRKD3 O94806 1/20 0.52
ABCB11 O95342 1/20 0.52
EGFR P00533 1/20 0.52
GBA1 P04062 1/20 0.52
NR3C1 P04150 1/20 0.52
ERBB2 P04626 1/20 0.52
PRKCG P05129 1/20 0.52
CYP1A2 P05177 1/20 0.52
PRKCB P05771 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1962745 0.87 ESR1 (0.59) ESR1ESR2MAPTCYP3A4MEN1
SCHEMBL227233 0.87 ESR1 (0.59) ESR1ESR2MAPTCYP3A4MEN1
SCHEMBL10506428 0.82 ESR1 (0.65) ESR1ESR2MAPTCYP3A4MEN1
SCHEMBL3773026 0.82 ESR1 (0.65) ESR1ESR2MAPTCYP3A4MEN1
SCHEMBL10506418 0.82 ESR1 (0.65) ESR1ESR2MAPTCYP3A4MEN1
SCHEMBL6673796 0.82 ESR1 (0.44) ESR1ESR2MAPTCYP3A4MEN1
SCHEMBL10379660 0.77 CYP19A1 (0.58) ESR1ESR2MAPTCYP3A4MEN1
SCHEMBL30402721 0.76 ESR1 (0.62) ESR1ESR2MAPTCYP3A4MEN1
Citric Acid SCHEMBL10954226 0.75 ESR1 (0.68) ESR1ESR2MAPTCYP3A4MEN1
SCHEMBL7547715 0.74 ESR1 (0.60) ESR1ESR2MAPTCYP3A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110698481-B Heteroaryl pyridone and aza-pyridone amide compounds 豪夫迈·罗氏有限公司 2023-02-28 CN disclosed