SCHEMBL3029604

SCHEMBL3029604

Brc1ccc2ncc(Br)n2c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAP3K14 Q99558 1/20 0.49
PIK3CA P42336 2/20 0.45
MTOR P42345 2/20 0.45
TSHR P16473 1/20 0.44
MAPK10 P53779 1/20 0.44
FLT3 P36888 1/20 0.40
PIK3CG P48736 1/20 0.38
GAA P10253 1/20 0.38
AHR P35869 2/20 0.35
ADORA2A P29274 1/20 0.34
PARP1 P09874 1/20 0.34
TRIM33 Q9UPN9 3/20 0.34
TRIM24 O15164 2/20 0.34
SCN10A Q9Y5Y9 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
MET P08581 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30217954 0.79 MAP3K14 (0.40) MAP3K14PIK3CAMTORPIK3CGSCN10A
SCHEMBL13676388 0.79 CYP1A2 (0.53) MAP3K14GAACYP1A2CYP2C9
SCHEMBL18785529 0.79 MAP3K14 (0.50) MAP3K14PIK3CAMTORTSHRMAPK10
SCHEMBL18041661 0.79 PIK3CA (0.47) MAP3K14PIK3CAMTORTSHRMAPK10
SCHEMBL3026036 0.79 MAP3K14 (0.33) MAP3K14PIK3CAMTORSCN10ACYP1A2
SCHEMBL381224 0.79 MAP3K14 (0.46) MAP3K14PIK3CAMTORTSHRMAPK10
SCHEMBL4821898 0.79 MAP3K14 (0.54) MAP3K14PIK3CAMTORTSHRMAPK10
SCHEMBL12998303 0.79 PIK3CA (0.47) MAP3K14PIK3CAMTORTSHRMAPK10
SCHEMBL22125606 0.79 MAP3K14 (0.50) MAP3K14PIK3CAMTORTSHRMAPK10
SCHEMBL3020269 0.79 POLB (0.51) MAP3K14FLT3AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114989167-B 3,6-dibromo or 3-bromoimidazo [1,2-a ] pyridine derivative and synthesis method thereof 江苏师范大学 2023-08-22 CN claimed
CN-114989167-A 3,6-dibromo or 3-bromo imidazo [1,2-a ] pyridine derivative and synthesis method thereof 江苏师范大学 2022-09-02 CN claimed
CN-114989167-B 3,6-dibromo or 3-bromoimidazo [1,2-a ] pyridine derivative and synthesis method thereof 江苏师范大学 2023-08-22 CN disclosed
CN-114989167-A 3,6-dibromo or 3-bromo imidazo [1,2-a ] pyridine derivative and synthesis method thereof 江苏师范大学 2022-09-02 CN disclosed
CN-105037356-A Synthesis method of 3,6-dibromoimidazole[1,2-a]pyridine SHANDONG YOUBANG BIOCHEMICAL TECHNOLOGY CO LTD 2015-11-11 CN disclosed
CN-105037356-A Synthesis method of 3,6-dibromoimidazole[1,2-a]pyridine SHANDONG YOUBANG BIOCHEMICAL TECHNOLOGY CO LTD 2015-11-11 CN disclosed
US-8367662-B2 Organic compounds NOVARTIS AG (CH) 2013-02-05 US disclosed
EP-2212323-B1 IMIDAZO [1,2-A] PYRIDINE DERIVATIVES USEFUL AS ALK INHIBITORS NOVARTIS AG (CH) 2012-08-15 EP disclosed
US-20100210641-A1 Organic Compounds NOVARTIS AG (CH) 2010-08-19 US disclosed
EP-2212323-A2 IMIDAZO [1,2-A] PYRIDINE DERIVATIVES USEFUL AS ALK INHIBITORS Novartis AG (CH) 2010-08-04 EP disclosed
WO-2009050183-A2 IMIDAZO [1, 2-A] PYRIDINE DERIVATIVES USEFUL AS ALK INHIBITORS NOVARTIS AG (CH) 2009-04-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100210641-A1 Organic Compounds ALK, ACVR1, ACVRL1 MAP3K14 1681/4885PIK3CA 741/4885MTOR 1367/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.