SCHEMBL30296171

SCHEMBL30296171

CCOC(=O)c1nc(-c2cccc(Cl)c2Cl)c(C)nc1N1CCC2(CC1)CO[C@@H](C)[C@H]2N

nearest known ligand 0.72

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 20/20 0.72
KCNH2 Q12809 2/20 0.72
EGFR P00533 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30511927 1.00 PTPN11 (0.72) PTPN11KCNH2EGFR
SCHEMBL26981010 1.00 PTPN11 (0.72) PTPN11KCNH2EGFR
SCHEMBL19785506 1.00 PTPN11 (0.72) PTPN11KCNH2EGFR
SCHEMBL21154556 0.84 PTPN11 (1.00) PTPN11KCNH2EGFR
SCHEMBL29374178 0.84 PTPN11 (1.00) PTPN11KCNH2EGFR
SCHEMBL25094875 0.84 PTPN11 (1.00) PTPN11KCNH2EGFR
SCHEMBL30295961 0.84 PTPN11 (1.00) PTPN11KCNH2EGFR
SCHEMBL21154462 0.84 PTPN11 (1.00) PTPN11KCNH2EGFR
SCHEMBL21154418 0.84 PTPN11 (1.00) PTPN11KCNH2EGFR
SCHEMBL29478950 0.84 PTPN11 (1.00) PTPN11KCNH2EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109983001-B 2, 5-disubstituted 3-methylpyrazines and 2,5, 6-trisubstituted 3-methylpyrazines as allosteric SHP2 inhibitors 锐新医药公司 2023-04-04 CN disclosed