SCHEMBL3029673

SCHEMBL3029673

Fc1ccc(-c2cc(-c3cnc4cc(-c5cccnc5)ccn34)ccn2)cc1

nearest known ligand 0.61

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 9/20 0.61
KDR P35968 6/20 0.61
GABRG2 P18507 1/20 0.57
GABRB3 P28472 1/20 0.57
GABRA3 P34903 1/20 0.57
FYN P06241 1/20 0.51
FGFR3 P22607 4/20 0.51
PIK3CA P42336 2/20 0.48
MTOR P42345 2/20 0.48
NEK2 P51955 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3029030 0.91 KDR (0.74) FLT3KDRGABRG2GABRB3GABRA3
SCHEMBL3028725 0.90 KDR (0.60) FLT3KDRGABRG2GABRB3GABRA3
SCHEMBL3024955 0.89 FLT3 (0.63) FLT3KDRFGFR3
SCHEMBL3025605 0.87 KDR (0.57) FLT3KDRGABRG2GABRB3GABRA3
SCHEMBL3328696 0.87 KDR (0.80) FLT3KDRGABRG2GABRB3GABRA3
SCHEMBL3020611 0.87 FLT3 (0.55) FLT3KDRGABRG2GABRB3GABRA3
SCHEMBL3021128 0.86 FLT3 (0.60) FLT3KDRFYNFGFR3
SCHEMBL3032703 0.85 KDR (0.62) FLT3KDRGABRG2GABRB3GABRA3
SCHEMBL3032412 0.83 FLT3 (0.59) FLT3KDRGABRG2GABRB3GABRA3
SCHEMBL3032518 0.83 FLT3 (0.62) FLT3KDRGABRG2GABRB3GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8367662-B2 Organic compounds NOVARTIS AG (CH) 2013-02-05 US disclosed
EP-2212323-B1 IMIDAZO [1,2-A] PYRIDINE DERIVATIVES USEFUL AS ALK INHIBITORS NOVARTIS AG (CH) 2012-08-15 EP disclosed
US-20100210641-A1 Organic Compounds NOVARTIS AG (CH) 2010-08-19 US disclosed
EP-2212323-A2 IMIDAZO [1,2-A] PYRIDINE DERIVATIVES USEFUL AS ALK INHIBITORS Novartis AG (CH) 2010-08-04 EP disclosed
WO-2009050183-A2 IMIDAZO [1, 2-A] PYRIDINE DERIVATIVES USEFUL AS ALK INHIBITORS NOVARTIS AG (CH) 2009-04-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100210641-A1 Organic Compounds ALK, ACVR1, ACVRL1 FLT3 4384/4885KDR 372/4885GABRG2 2020/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.