SCHEMBL30317153

SCHEMBL30317153

[2H]N1C(=O)Cc2cc(OC)c(OC(C)C)cc2C1c1ccc(Cl)cc1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 19/20 0.56
MDM4 O15151 14/20 0.56
CRHBP P24387 1/20 0.47
CRHR2 Q13324 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30225606 0.89 CRHBP (0.58) MDM2MDM4CRHBPCRHR2
SCHEMBL30225589 0.89 CRHBP (0.58) MDM2MDM4CRHBPCRHR2
SCHEMBL2395864 0.89 CRHBP (0.58) MDM2MDM4CRHBPCRHR2
SCHEMBL2393838 0.89 CRHBP (0.58) MDM2MDM4CRHBPCRHR2
SCHEMBL30225612 0.89 CRHBP (0.58) MDM2MDM4CRHBPCRHR2
SCHEMBL23842064 0.89 CRHBP (0.58) MDM2MDM4CRHBPCRHR2
SCHEMBL15701400 0.84 MDM2 (0.50) MDM2MDM4CRHBPCRHR2
SCHEMBL15701402 0.84 MDM2 (0.50) MDM2MDM4CRHBPCRHR2
SCHEMBL12258915 0.84 MDM2 (0.50) MDM2MDM4CRHBPCRHR2
SCHEMBL10854785 0.80 CRHBP (0.67) MDM2MDM4CRHBPCRHR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115776887-A MDM2 degrading agents and uses thereof 凯麦拉医疗公司 2023-03-10 CN disclosed